Azido-mono-amide-DOTA

Name: Azido-mono-amide-DOTA
Brand: MedChemExpress
SKU: HY-W539916
Rating: 4.5 (1 reviews)

Cat. No.: HY-W539916 Purity: 99.96%: FAQs
Data Sheet SDS COA Handling Instructions Technical Support

Azido-mono-amide-DOTAis a bifunctional chelator (Bifunctional Chelator; BFC) and a macrocyclic DOTA derivative used for tumor pre-targeting. Azido-mono-amide-DOTA can be used for conjugation of peptides and radionuclides.

For research use only. We do not sell to patients.

Azido-mono-amide-DOTA Chemical Structure

CAS No. : 1227407-76-2

Size	Stock	Quantity
10 mg	In-stock	Estimated Time of Arrival: December 31
50 mg	Get quote
100 mg	Get quote

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Customer Review

Based on 1 publication(s) in Google Scholar

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•Related Small Molecules:

•Related Proteins:

View All Radionuclide-Drug Conjugates (RDCs) Isoform Specific Products:

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RDC Peptide RDC Antibody RDC Bifunctional Chelator RDC Linker Other

Biological Activity
Purity & Documentation
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Description

IC₅₀ & Target

RDC Bifunctional Chelator

Molecular Weight

486.52

Formula

C₁₉H₃₄N₈O₇

CAS No.

1227407-76-2

Appearance

Solid

Color

White to off-white

SMILES

[N-]=[N+]=NCCCNC(CN1CCN(CCN(CCN(CC1)CC(O)=O)CC(O)=O)CC(O)=O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Powder	-20°C	3 years
	4°C	2 years
In solvent	-80°C	6 months
	-20°C	1 month

Solvent & Solubility

In Vitro:

H₂O : ≥ 100 mg/mL (205.54 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	2.0554 mL	10.2771 mL	20.5541 mL
5 mM	0.4111 mL	2.0554 mL	4.1108 mL
10 mM	0.2055 mL	1.0277 mL	2.0554 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.

Molarity Calculator
Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Concentration _(start)

Volume _(start)

Concentration _(final)

Volume _(final)

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

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μL

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

This product has good water solubility, please refer to the measured solubility data in water/PBS/Saline for details.

The concentration of the stock solution you require exceeds the measured solubility. The following solution is for reference only.If necessary, please contact MedChemExpress (MCE).

Purity & Documentation

Purity: 99.96%

Select Batch:

Data Sheet (242 KB) SDS (251 KB)

COA (247 KB) HNMR (270 KB) RP-HPLC (235 KB) MS (68 KB)

Handling Instructions (2659 KB)

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

H₂O	1 mM	2.0554 mL	10.2771 mL	20.5541 mL	51.3854 mL
	5 mM	0.4111 mL	2.0554 mL	4.1108 mL	10.2771 mL
	10 mM	0.2055 mL	1.0277 mL	2.0554 mL	5.1385 mL
	15 mM	0.1370 mL	0.6851 mL	1.3703 mL	3.4257 mL
	20 mM	0.1028 mL	0.5139 mL	1.0277 mL	2.5693 mL
	25 mM	0.0822 mL	0.4111 mL	0.8222 mL	2.0554 mL
	30 mM	0.0685 mL	0.3426 mL	0.6851 mL	1.7128 mL
	40 mM	0.0514 mL	0.2569 mL	0.5139 mL	1.2846 mL
	50 mM	0.0411 mL	0.2055 mL	0.4111 mL	1.0277 mL
	60 mM	0.0343 mL	0.1713 mL	0.3426 mL	0.8564 mL
	80 mM	0.0257 mL	0.1285 mL	0.2569 mL	0.6423 mL
	100 mM	0.0206 mL	0.1028 mL	0.2055 mL	0.5139 mL

* Note: If you choose water as the stock solution, please dilute it to the working solution, then filter and sterilize it with a 0.22 μm filter before use.