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Results for "

β-adrenergic

" in MedChemExpress (MCE) Product Catalog:

By Targets:	Adrenergic Receptor (128) 5-HT Receptor (5) Antibiotic (1) Autophagy (5) Bacterial (4) Calcium Channel (3) Cytochrome P450 (3) Endogenous Metabolite (11) iGluR (4) Isotope-Labeled Compounds (9) mAChR (4) Melanocortin Receptor (1) Mitophagy (2) P2X Receptor (2) Phosphodiesterase (PDE) (1) Potassium Channel (4) Prostaglandin Receptor (1) Small Interfering RNA (siRNA) (2) Sodium Channel (3) TRP Channel (1)
By Research Areas:	Cancer (5) Cardiovascular Disease (76) Endocrinology (55) Infection (2) Inflammation/Immunology (15) Metabolic Disease (6) Neurological Disease (32)
Click Chemistry:	Alkynes (1)
Oligonucleotides:	siRNAs (2)

138

Inhibitors & Agonists

Peptides

Natural
Products

Isotope-Labeled Compounds

Click Chemistry

Oligonucleotides

Targets Recommended: Adrenergic Receptor

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-102032

Butyryltimolol	Adrenergic Receptor	Endocrinology
Butyryltimolol, an effective precursor of Timolol, improves the corneal penetration of Timolol . Butyryltimolol is a *β-adrenergic* blocker .

HY-102032A

(RS)-Butyryltimolol	Adrenergic Receptor	Others
(RS)-Butyryltimolol is the racemate of Butyryltimolol. Butyryltimolol, an effective proagent of Timolol, improves the corneal penetration of Timolol . Butyryltimolol is a β-adrenergic blocker .

HY-N0132A

Synephrine hydrochloride Oxedrine hydrochloride	Adrenergic Receptor Endogenous Metabolite	Neurological Disease Endocrinology
Synephrine (Oxedrine) hydrochloride, an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine hydrochloride is a sympathomimetic compound and can be used for weight loss .

HY-N0132

Synephrine Oxedrine	Adrenergic Receptor Endogenous Metabolite	Neurological Disease Endocrinology
Synephrine (Oxedrine), an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine is a sympathomimetic compound and can be used for weight loss .

HY-105154A

Proxodolol	Adrenergic Receptor	Cardiovascular Disease
Proxodolol is a β-adrenergic receptor blocker. Proxodolol can be used for the study of arterial hypertension .

HY-113797

RS-52367	Adrenergic Receptor	Others
RS-52367 is a potent syntex *β-adrenergic* antagonist. RS-52367 decreases intraocular pressure with a mild systemic effect in dogs .

HY-120519

L-665871	Adrenergic Receptor	Metabolic Disease
L-665871 is a orally active β-adrenergic receptor agonist that can be used as a swine growth promoter .

HY-N0132B

Synephrine hemitartrate Oxedrine hemitartrate	Adrenergic Receptor Endogenous Metabolite	Neurological Disease
Synephrine (Oxedrine) hemitartrate, an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine hemitartrate is a sympathomimetic compound and can be used for weight loss .

HY-107010A

Esprolol hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Esprolol (hydrochloride) is an orally active and potent β-adrenergic receptor antagonist. Esprolol (hydrochloride) undergoes rapid metabolism by blood and tissue esterases to form an active metabolite, amoxolol. Esprolol (hydrochloride) is promising for research of exertional angina .

HY-121082

(-)-Dihydroalprenolol L-Dihydroalprenolol	Others	Endocrinology
(-)-Dihydroalprenolol (L-Dihydroalprenolol) is a β-adrenergic antagonist that inhibits the activity of β-adrenergic receptors. (-)-Dihydroalprenolol can cause desensitization of approximately 60% of β-adrenergic receptor binding sites. (-)-Dihydroalprenolol has also been shown to reduce the binding capacity of specific β-adrenergic ligands. (-)-Dihydroalprenolol may affect the ability to stimulate membrane-bound adenylate acylase .

HY-N0132R

Synephrine (Standard) Oxedrine (Standard)	Adrenergic Receptor Endogenous Metabolite	Endocrinology
Synephrine (Standard) is the analytical standard of Synephrine. This product is intended for research and analytical applications. Synephrine (Oxedrine), an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine is a sympathomimetic compound and can be used for weight loss .

HY-N0132AR

Synephrine hydrochloride (Standard)	Adrenergic Receptor Endogenous Metabolite	Neurological Disease Endocrinology
Synephrine (hydrochloride) (Standard) is the analytical standard of Synephrine (hydrochloride). This product is intended for research and analytical applications. Synephrine (Oxedrine) hydrochloride, an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine hydrochloride is a sympathomimetic compound and can be used for weight loss .

HY-122364

Bucumolol hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Bucumolol hydrochloride is a β-adrenergic receptor antagonist that can slow heart rate (negative chronotropic effect) and reduce cardiac contractility (negative inotropic effect). Bucumolol hydrochloride has antiarrhythmic and local anesthetic activity and can be used in the study of cardiovascular diseases .

HY-U00016

Teoprolol	Adrenergic Receptor	Endocrinology
Teoprolol is a β-adrenergic receptor blocker.

HY-131105

Cimbuterol	Adrenergic Receptor	Cardiovascular Disease Endocrinology
Cimbuterol is a β-adrenergic receptor agonist .

HY-101585

Imoxiterol RP 58802B	Adrenergic Receptor	Neurological Disease Endocrinology
Imoxiterol (RP 58802B) is a *β-adrenergic* agonist.

HY-131145

Brombuterol hydrochloride Bromobuterol hydrochloride	Adrenergic Receptor	Inflammation/Immunology
Brombuterol hydrochloride (Bromobuterol hydrochloride) is a β-adrenergic receptor agonist .

HY-B1481

Isoetharine mesylate Isoetarine mesylate	Adrenergic Receptor	Cardiovascular Disease Inflammation/Immunology
Isoetharine (Isoetarine) mesylate is an orally active selective agonist of β-adrenergic receptors. Isoetharine mesylate is a catechol-like agent and catechol O-methyltransferase (COMT) mediates its methylation. Isoetharine mesylate can promote the production of cAMP which stimulates the relaxation of smooth muscle cells and can be used as an emphysema, bronchitis and bronchodilator .

HY-B1481A

Isoetharine Isoetarine	Adrenergic Receptor	Cardiovascular Disease Inflammation/Immunology
Isoetharine (Isoetarine) is an orally active selective agonist of β-adrenergic receptors. Isoetharine is a catechol-like agent and catechol O-methyltransferase (COMT) mediates its methylation. Isoetharine can promote the production of cAMP which stimulates the relaxation of smooth muscle cells and can be used as an emphysema, bronchitis and bronchodilator .

HY-123012

Lubabegron LY-488756	Adrenergic Receptor	Others
Lubabegron is a potent modulator of β-adrenergic receptor (β -AR). Lubabegron demonstrates antagonistic behavior at the β₁ and β ₂ receptor subtypes and agonistic behavior at the β ₃ receptor subtype in cattle. Lubabegron reduces NH₃ gas emissions from an animal or its waste .

HY-B1694

Methoxyphenamine NSC-65644 free base	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Methoxyphenamine is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.

HY-B0804

Nadolol 1 Publications Verification SQ-11725	Adrenergic Receptor	Cardiovascular Disease
Nadolol (SQ-11725) is a non-selective and orally active β-adrenergic receptors blocker and is a substrate of organic anion transporting polypeptide 1A2 (OATP1A2). Nadolol has the the potential for high blood pressure, angina pectoris and vascular headaches research .

HY-U00283

Falintolol, (Z)-	Adrenergic Receptor	Endocrinology
Falintolol, (Z)-, a new *β-adrenergic* antagonist, is characterized by the presence of an oxime function.

HY-116888

BFE-55	Adrenergic Receptor	Endocrinology
BFE-55 is a derivative of befunolol and a β-adrenergic partial agonist .

HY-169137

Falintolol	Adrenergic Receptor	Others
Falintolol is a β-adrenergic receptor antagonist that can be used in glaucoma research .

HY-131103

Phenylethanolamine A	Adrenergic Receptor	Metabolic Disease Inflammation/Immunology
Phenylethanolamine A acts as a *β-adrenergic* agonist. Phenylethanolamine A is a byproduct during the Ractopamine synthesis process .

HY-B1694A

Methoxyphenamine hydrochloride NSC-65644	Adrenergic Receptor	Inflammation/Immunology Endocrinology
Methoxyphenamine hydrochloride, a non-regulated analog of Methamphetamine, is a β-adrenergic receptor agonist used as a bronchodilator .

HY-131105S

Cimbuterol-d9	Isotope-Labeled Compounds Adrenergic Receptor	Cardiovascular Disease
Cimbuterol-d₉ is the deuterium labeled Cimbuterol. Cimbuterol is aβ-adrenergic agonist[1].

HY-153483

Bamosiran SYL040012	Adrenergic Receptor Small Interfering RNA (siRNA)	Others
Bamosiran is a small interfering RNA targeting β-adrenergic receptor 2, and is used to lower intraocular pressure

HY-153483A

Bamosiran sodium SYL040012 sodium	Adrenergic Receptor Small Interfering RNA (siRNA)	Others
Bamosiran sodium is a small interfering RNA targeting β-adrenergic receptor 2, and is used to lower intraocular pressure

HY-B0804R

Nadolol (Standard)	Adrenergic Receptor	Cardiovascular Disease
Nadolol (Standard) is the analytical standard of Nadolol. This product is intended for research and analytical applications. Nadolol (SQ-11725) is a non-selective and orally active β-adrenergic receptors blocker and is a substrate of organic anion transporting polypeptide 1A2 (OATP1A2). Nadolol has the the potential for high blood pressure, angina pectoris and vascular headaches research .

HY-131104AS

Brombuterol-d9 hydrochloride Bromobuterol d₉ hydrochloride	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology
Brombuterol-d₉ (hydrochloride) is a deuterium labeled Brombuterol hydrochloride. Brombuterol hydrochloride is a β-adrenergic receptor agonist[1].

HY-131104S

Brombuterol-d9 Bromobuterol d₉	Isotope-Labeled Compounds Adrenergic Receptor	Inflammation/Immunology
Brombuterol-d₉ is a deuterium labeled Brombuterol. Brombuterol is a β-adrenergic receptor agonist[1].

HY-136449

Bromchlorbuterol hydrochloride	Adrenergic Receptor	Inflammation/Immunology
Bromchlorbuterol hydrochloride is an active β-adrenergic agonist (β-agonist) and can be used for the research of pulmonary disease and asthma .

HY-121005

Bufetolol	Adrenergic Receptor	Cardiovascular Disease
Bufetolol is an inhibitor for β-adrenergic receptor, that affects the maximum velocity of rise of the action potential, and exhibits antiarrhythmic efficacy .

HY-B0573S

Propranolol-d7 hydrochloride	Adrenergic Receptor	Cardiovascular Disease Neurological Disease Endocrinology
Propranolol-d₇ (hydrochloride) is a deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively[1]. Propranolol hydrochloride inhibits [3H]-DHA binding to rat brain membrane preparation with an IC50 of 12 nM[2]. Propranolol hydrochloride is used for the study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy[3].

HY-B2111

(R)-(+)-Atenolol	Adrenergic Receptor	Cardiovascular Disease Others
(R)-(+)-Atenolol is the less active enantiomer of the (R,S)-atenolol. (R,S)-atenolol is a β-adrenergic receptor antagonist .

HY-121567

Metipranolol 1 Publications Verification	Adrenergic Receptor	Cardiovascular Disease
Metipranolol is a nonselective and orally active β-adrenergic receptor antagonist. Metipranolol can be used for hypertension and glaucoma research .

HY-131145R

Brombuterol hydrochloride (Standard)	Adrenergic Receptor	Inflammation/Immunology
Brombuterol (hydrochloride) (Standard) is the analytical standard of Brombuterol (hydrochloride). This product is intended for research and analytical applications. Brombuterol hydrochloride (Bromobuterol hydrochloride) is a β-adrenergic receptor agonist .

HY-101656A

Medroxalol hydrochloride RMI81968 hydrochloride	Adrenergic Receptor	Cardiovascular Disease
Medroxalol hydrochloride is an orally active adrenergic receptor antagonist, blocks α- and β-adrenergic receptors. Medroxalol hydrochloride shows antihypertensive and vasodilating effects .

HY-B0804S

Nadolol-d9 SQ-11725-d₉	Adrenergic Receptor	Cardiovascular Disease Endocrinology
Nadolol-d₉ is the deuterium labeled Nadolol. Nadolol is a non-selective and orally active β-adrenergic receptors blocker[1].

HY-N10452

Methyl maslinate	Adrenergic Receptor	Cardiovascular Disease
Methyl maslinate is a *β-adrenergic* antagonist. Methyl maslinate is a potent cardiotonic and antidysrhythmic agent. Methyl maslinate has the potential for hypertension research .

HY-A0252A

Bupranolol hydrochloride	Others	Cancer
Bupranolol hydrochloride is a non-selective β-adrenergic blocker with potent membrane stabilizing activity. Bupranolol hydrochloride is able to significantly modulate the contractile activity of the non-pregnant human uterus. Bupranolol hydrochloride showed significant effects on spontaneous uterine contractions in an in vitro study in patients with ovarian cancer. Bupranolol hydrochloride is similar in potency to propranolol, another β-adrenergic blocker. Bupranolol hydrochloride is rapidly and completely absorbed in vivo, and its major metabolite is carboxybupranolol .

HY-101656

Medroxalol RMI81968	Adrenergic Receptor	Cardiovascular Disease
Medroxalol (RMI81968) is an orally active adrenergic receptor antagonist, blocks α- and β-adrenergic receptors. Medroxalol shows antihypertensive and vasodilating effects .

HY-119006

L-640,033	Adrenergic Receptor	Endocrinology
L-640,033 is a potent agonist of *β-adrenergic*. L-640,033 play an important role in lipid metabolism, and growth .

HY-108302

Nifenalol	Adrenergic Receptor	Others
Nifenalol is a β-adrenergic receptor blocker. Nifenalol inhibits β-adrenoceptor differentiation in right atrium, diaphragm and adipose tissue in a rat model .

HY-121185

Hexoprenaline	Adrenergic Receptor	Infection Inflammation/Immunology
Hexoprenaline is an orally active and selective β-adrenergic receptor agonist that dilates the bronchi. Hexoprenaline can be used in the study of bronchospasm, including asthma, bronchitis, and emphysema .

HY-B1392A

Esmolol	Adrenergic Receptor	Cardiovascular Disease
Esmolol is a potent and cardio-selective *β-adrenergic* blocker. Esmolol shows cardioprotection. Esmolol has the potential for the research of tachycardia with ischemic heart disease .

HY-131103S

Phenylethanolamine A-d3	Adrenergic Receptor	Metabolic Disease Inflammation/Immunology
Phenylethanolamine A-d₃ is a deuterium labeled Phenylethanolamine A. Phenylethanolamine A acts as a β-adrenergic agonist. Phenylethanolamine A is a byproduct during the Ractopamine synthesis process[1].

HY-B1486

Oxprenolol hydrochloride 1 Publications Verification Ba 39089	Adrenergic Receptor	Cardiovascular Disease
Oxprenolol hydrochloride (Ba 39089) is an orally bioavailable *β-adrenergic* receptor (β-AR) antagonist with a K_i of 7.10 nM in a radioligand binding assay using rat heart muscle .

Cat. No.	Product Name	Target	Research Area

HY-P1376A

G-Protein antagonist peptide TFA	mAChR Adrenergic Receptor	Endocrinology
G-Protein antagonist peptide TFA is a truncated substance P-related peptide, competes with receptor for G protein binding. G-Protein antagonist peptide TFA inhibits the activation of G_i or G_o by M2 muscarinic cholinergic receptor (M2 mAChR) or of G_s by beta-adrenergic receptor in the reconstituted phospholipid vesicles, assayed by receptor-promoted GTP hydrolysis .

HY-P10336

Serpinin	Peptides	Neurological Disease Endocrinology
Serpinin is an agonist of the protease inhibitor Nexin-1 (PN-1). Serpinin upregulates the expression of PN-1 through the cAMP-PKA-Sp1 signaling pathway, promoting granule biogenesis in endocrine cells. Serpinin is used in research related to the regulation of secretory function . Serpinin is a selective agonist for β-adrenergic receptors. Serpinin interacts with β1-adrenergic receptors to activate the AC-cAMP-PKA pathway, which regulates myocardial systolic and diastolic function. pGlu-serpinin upregulates Bcl2 mRNA transcription and exerts neuroprotective effects .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-N0132A

Synephrine hydrochloride Oxedrine hydrochloride	Structural Classification Citrus × aurantium Linnaeus Neurological Disease Classification of Application Fields Source classification Rutaceae Plants Endogenous metabolite Alkaloids Monophenols Other Alkaloids Phenols Disease Research Fields Endocrinology	Adrenergic Receptor Endogenous Metabolite
Synephrine (Oxedrine) hydrochloride, an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine hydrochloride is a sympathomimetic compound and can be used for weight loss .

HY-N0132

Synephrine Oxedrine	Structural Classification Citrus × aurantium Linnaeus Neurological Disease Classification of Application Fields Rutaceae Plants Endogenous metabolite Alkaloids Monophenols Other Alkaloids Phenols Disease Research Fields Endocrinology	Adrenergic Receptor Endogenous Metabolite
Synephrine (Oxedrine), an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine is a sympathomimetic compound and can be used for weight loss .

HY-B2111

(R)-(+)-Atenolol	Cardiovascular Disease Classification of Application Fields Disease Research Fields	Adrenergic Receptor
(R)-(+)-Atenolol is the less active enantiomer of the (R,S)-atenolol. (R,S)-atenolol is a β-adrenergic receptor antagonist .

HY-B1035

Levobunolol hydrochloride 1 Publications Verification l-Bunolol hydrochloride	Cardiovascular Disease Classification of Application Fields Disease Research Fields	Adrenergic Receptor
Levobunolol (l-Bunolol) hydrochloride is a potent and nonselective β-adrenergic receptor antagonist. Levobunolol hydrochloride is an ocular hypotensive agent and lowers mean intraocular pressure (IOP). Levobunolol hydrochloride can be used for glaucoma and superior oblique myokymia (SOM) research .

HY-B0468

Isoprenaline hydrochloride Maximum Cited Publications 51 Publications Verification Isoproterenol hydrochloride	Cardiovascular Disease Structural Classification Alkaloids Classification of Application Fields Other Alkaloids Source classification Phenols Polyphenols Endogenous metabolite Disease Research Fields Endocrinology	Adrenergic Receptor Endogenous Metabolite
Isoprenaline (Isoproterenol) hydrochloride is a non-selective, orally active β-adrenergic receptor agonist. Isoprenaline has potent peripheral vasodilator, bronchodilator, and cardiac stimulating activities. Isoprenaline can be used for the research of bradycardia and bronchial asthma .

HY-N0132B

Synephrine hemitartrate Oxedrine hemitartrate	Alkaloids Monophenols Source classification Rutaceae Phenols Plants Citrus reticulata Blanco	Adrenergic Receptor Endogenous Metabolite
Synephrine (Oxedrine) hemitartrate, an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine hemitartrate is a sympathomimetic compound and can be used for weight loss .

HY-N0132R

Synephrine (Standard) Oxedrine (Standard)	Structural Classification Alkaloids Citrus × aurantium Linnaeus Neurological Disease Classification of Application Fields Source classification Rutaceae Phenols Plants Endogenous metabolite Disease Research Fields Endocrinology	Adrenergic Receptor Endogenous Metabolite
Synephrine (Standard) is the analytical standard of Synephrine. This product is intended for research and analytical applications. Synephrine (Oxedrine), an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine is a sympathomimetic compound and can be used for weight loss .

HY-N0132AR

Synephrine hydrochloride (Standard)	Alkaloids Structural Classification Citrus × aurantium Linnaeus Monophenols Other Alkaloids Source classification Rutaceae Phenols Plants Endogenous metabolite	Adrenergic Receptor Endogenous Metabolite
Synephrine (hydrochloride) (Standard) is the analytical standard of Synephrine (hydrochloride). This product is intended for research and analytical applications. Synephrine (Oxedrine) hydrochloride, an alkaloid, is an *α-adrenergic* and *β-adrenergic* agonist derived from the Citrus aurantium. Synephrine hydrochloride is a sympathomimetic compound and can be used for weight loss .

HY-N10452

Methyl maslinate	Natural Products Source classification Rosaceae Plants Eriobotrya japonica (Thunb.) Lindl.	Adrenergic Receptor
Methyl maslinate is a *β-adrenergic* antagonist. Methyl maslinate is a potent cardiotonic and antidysrhythmic agent. Methyl maslinate has the potential for hypertension research .

HY-108353

Isoprenaline	Cardiovascular Disease Structural Classification Alkaloids Classification of Application Fields Other Alkaloids Source classification Phenols Polyphenols Endogenous metabolite Disease Research Fields Endocrinology	Adrenergic Receptor Endogenous Metabolite
Isoprenaline is a non-selective, orally active β-adrenergic receptor agonist. Isoprenaline has potent peripheral vasodilator, bronchodilator, and cardiac stimulating activities. Isoprenaline can be used for the research of bradycardia and bronchial asthma .

HY-108353A

Isoprenaline hemisulfate	Cardiovascular Disease Structural Classification Alkaloids Classification of Application Fields Other Alkaloids Source classification Phenols Polyphenols Endogenous metabolite Disease Research Fields Endocrinology	Adrenergic Receptor Endogenous Metabolite
Isoprenaline hemisulfate is a non-selective, orally active β-adrenergic receptor agonist. Isoprenaline has potent peripheral vasodilator, bronchodilator, and cardiac stimulating activities. Isoprenaline can be used for the research of bradycardia and bronchial asthma .

HY-B0468R

Isoprenaline hydrochloride (Standard)	Structural Classification Alkaloids Other Alkaloids Source classification Phenols Polyphenols Endogenous metabolite	Adrenergic Receptor Endogenous Metabolite
Isoprenaline (hydrochloride) (Standard) is the analytical standard of Isoprenaline (hydrochloride). This product is intended for research and analytical applications. Isoprenaline (Isoproterenol) hydrochloride is a non-selective, orally active β-adrenergic receptor agonist. Isoprenaline has potent peripheral vasodilator, bronchodilator, and cardiac stimulating activities. Isoprenaline can be used for the research of bradycardia and bronchial asthma .

HY-B0573

Propranolol hydrochloride 20+ Cited Publications	Alkaloids Neurological Disease Classification of Application Fields Other Alkaloids Source classification Endogenous metabolite Disease Research Fields Endocrinology	Adrenergic Receptor Bacterial
Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with K_i values of 1.8 nM and 0.8 nM, respectively . Propranolol hydrochloride inhibits [ ³H]-DHA binding to rat brain membrane preparation with an IC₅₀ of 12 nM . Propranolol hydrochloride is used for study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy .

HY-B0573B

Propranolol 20+ Cited Publications	Cardiovascular Disease Alkaloids Neurological Disease Classification of Application Fields Source classification Endogenous metabolite Disease Research Fields	Adrenergic Receptor Bacterial
Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with K_i values of 1.8 nM and 0.8 nM, respectively . Propranolol inhibits [ ³H]-DHA binding to rat brain membrane preparation with an IC₅₀ of 12 nM . Propranolol is used for the study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy .

HY-B0573R

Propranolol hydrochloride (Standard)	Alkaloids Other Alkaloids Source classification Endogenous metabolite	Adrenergic Receptor Bacterial
Propranolol (hydrochloride) (Standard) is the analytical standard of Propranolol (hydrochloride). This product is intended for research and analytical applications. Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with K_i values of 1.8 nM and 0.8 nM, respectively . Propranolol hydrochloride inhibits [ ³H]-DHA binding to rat brain membrane preparation with an IC₅₀ of 12 nM . Propranolol hydrochloride is used for study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy .

HY-108306

Moprolol (±)-Moprolol	Cardiovascular Disease Classification of Application Fields Disease Research Fields	Adrenergic Receptor
Moprolol ((±)-Moprolol) is an beta-adrenergic receptor blocker, which can be used for research in essential hypertension .

Cat. No.	Product Name	Chemical Structure

HY-131104S

Brombuterol-d9
Brombuterol-d₉ is a deuterium labeled Brombuterol. Brombuterol is a β-adrenergic receptor agonist[1].

HY-B0573S

Propranolol-d7 hydrochloride

Propranolol-d₇ (hydrochloride) is a deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively[1]. Propranolol hydrochloride inhibits [3H]-DHA binding to rat brain membrane preparation with an IC50 of 12 nM[2]. Propranolol hydrochloride is used for the study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy[3].

HY-B0804S

Nadolol-d9
Nadolol-d₉ is the deuterium labeled Nadolol. Nadolol is a non-selective and orally active β-adrenergic receptors blocker[1].

HY-131103S

Phenylethanolamine A-d3
Phenylethanolamine A-d₃ is a deuterium labeled Phenylethanolamine A. Phenylethanolamine A acts as a β-adrenergic agonist. Phenylethanolamine A is a byproduct during the Ractopamine synthesis process[1].

HY-B1486S

Oxprenolol-d7 hydrochloride
Oxprenolol-d₇ (hydrochloride) is the deuterium labeled Oxprenolol hydrochloride. Oxprenolol hydrochloride (Ba 39089) is an orally bioavailable β-adrenergic receptor (β-AR) antagonist with a Ki of 7.10 nM in a radioligand binding assay using rat heart muscle[1].

HY-B0437AS

Sotalol-d6 hydrochloride
Sotalol-d₆ (hydrochloride) is a deuterium labeled Sotalol hydrochloride. Sotalol hydrochloride is an orally active, non-selective competitive β-adrenergic receptor blocker. Sotalol hydrochloride is a potent antiarrhythmic agent that can be used for the research of pediatric arrhythmias. Sotalol hydrochloride blocks β-receptors, and potassium KCNH2 channels[1][2].

HY-131105S

Cimbuterol-d9
Cimbuterol-d₉ is the deuterium labeled Cimbuterol. Cimbuterol is aβ-adrenergic agonist[1].

HY-131104AS

Brombuterol-d9 hydrochloride
Brombuterol-d₉ (hydrochloride) is a deuterium labeled Brombuterol hydrochloride. Brombuterol hydrochloride is a β-adrenergic receptor agonist[1].

HY-B1486AS

Oxprenolol-d7
Oxprenolol-d₇ is the deuterium labeled Oxprenolol. Oxprenolol (Ba 39089 free base) is an orally bioavailable β-adrenergic receptor (β-AR) antagonist with a Ki of 7.10 nM in a radioligand binding assay using rat heart muscle[1].

HY-B0468S

Isoprenaline-d7 hydrochloride
Isoprenaline-d7 (hydrochloride) is a deuterated labeled Isoprenaline (hydrochloride) . Isoprenaline (Isoproterenol) hydrochloride is a non-selective, orally active β-adrenergic receptor agonist. Isoprenaline has potent peripheral vasodilator, bronchodilator, and cardiac stimulating activities. Isoprenaline can be used for the research of bradycardia and bronchial asthma .

HY-B0437S

Sotalol-d6
Sotalol-d₆ is the deuterium labeled Sotalol. Sotalol is an orally active, non-selective β-adrenergic receptor blocker. Sotalol is a potent antiarrhythmic agent that can be used for the research of pediatric arrhythmias. Sotalol blocks β-receptors, and potassium KCNH2 channels. Antiepileptic Agent[1][2][3][4].

HY-W728545

Labetalol-d6 hydrochloride
Labetalol-d6 hydrochloride (AH5158-d6 hydrochloride; Sch-15719W-d6) is a deuterium labeled Labetalol (HY-121383). Labetalol is an orally active α1- and β-adrenergic receptors competitive antagonist, which exhibits anti-hypertensive property .

HY-100935S

Cimaterol-d7
Cimaterol-d₇ is the deuterium labeled Cimaterol. Cimaterol is a potent agonist of β-adrenergic receptors (pEC50s=8.13, 8.78, and 6.62 for human β1, β2, and β3, respectively). Cimaterol has been used in farmed animals to increase carcass mass and to alter muscle and fat deposition.

HY-A0016S

Dronedarone D6 hydrochloride

Dronedarone-d₆ (hydrochloride) is the deuterium labeled Dronedarone. Dronedarone hydrochloride, a derivative of Amiodarone (HY-14187), is a class III antiarrhythmic agent for the study of atrial fibrillation (AF) and atrial flutter. Dronedarone hydrochloride is a potent blocker of multiple ion currents, including potassium current, sodium current, and L-type calcium current, and exhibits antiadrenergic effects by noncompetitive binding to β-adrenergic receptors. Dronedarone hydrochloride is a substrate for and a moderate inhibitor of CYP3A4[1][2][3][4].

HY-B0573BS

Propranolol-d7

Propranolol-d₇ is the deuterium labeled Propranolol. Propranolol is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively[1]. Propranolol inhibits [3H]-DHA binding to rat brain membrane preparation with an IC50 of 12 nM[2]. Propranolol is used for the study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy[3].

HY-B1270S

Isoxsuprine-d6 hydrochloride
Isoxsuprine-d₆ (hydrochloride) is the deuterium labeled Isoxsuprine hydrochloride. Isoxsuprine hydrochloride is a beta-adrenergic receptor agonist with Kis of 13.65 μΜ and 3.48 μΜ for myometrial and placcntal beta-adrenergic receptor, respectively. Isoxsuprine hydrochloride is also a NMDA receptor antagonist.

HY-B0573S1

Propranolol-d7 (ring-d7)

Propranolol-d₇ (ring-d₇) is the deuterium labeled Propranolol hydrochloride. Propranolol hydrochloride is a nonselective β-adrenergic receptor (βAR) antagonist, has high affinity for the β1AR and β2AR with Ki values of 1.8 nM and 0.8 nM, respectively[1]. Propranolol hydrochloride inhibits [3H]-DHA binding to rat brain membrane preparation with an IC50 of 12 nM[2]. Propranolol hydrochloride is used for study of hypertension, pheochromocytoma, myocardial infarction, cardiac arrhythmias, angina pectoris, and hypertrophic cardiomyopathy[3].

HY-B1392S

Esmolol-d7 hydrochloride
Esmolol-d₇ (hydrochloride) is the deuterium labeled Esmolol hydrochloride. Esmolol hydrochloride is a beta adrenergic receptor blocker[1][2].

HY-B0982S

Pindolol-d7
Pindolol-d₇ (LB-46-d7) is the deuterium labeled Pindolol. Pindolol (LB-46) is a nonselective β-blocker with partial beta-adrenergic receptor agonist activity, also functions as a 5-HT1A receptor weak partial antagonist (Ki=33 nM)[1][2].

Cat. No.	Product Name		Classification

HY-101658

Pargolol hydrochloride Ko 1400 hydrochloride		Alkynes
Pargolol hydrochloride is a β adrenergic receptor antagonist. Pargolol hydrochloride is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.

Cat. No.	Product Name		Classification