1. Signaling Pathways
  2. Anti-infection
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  4. HIV Inhibitors

HIV Inhibitors

HIV

HIV-1

HIV-2

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HIV Inhibitors, Antagonists & Activators
Product Name HIV HIV-1 HIV-2 Purity
Chloroquine  
HIV-1
  99.82%
Doxorubicin hydrochloride  
HIV-1
  99.90%
5-Fluorouracil
HIV
    99.99%
Chloroquine phosphate  
HIV-1
  99.89%
Panobinostat  
HIV-1
 
Hydroxyurea  
HIV-1
  ≥98.0%
Plerixafor  
HIV-1, EC50: 1-10 nM
HIV-2, EC50: 1-10 nM
98.61%
Maraviroc  
HIV-1 (Ba-L), IC50: 1.1 nM (in PM-1 cells)
  99.88%
Ivermectin  
HIV-1
  98.01%
Ebselen  
HIV-1
  99.58%
Plerixafor octahydrochloride  
HIV-1, EC50: 1-10 nM
HIV-2, EC50: 1-10 nM
≥98.0%
CK-666  
HIV-1
  99.17%
Rottlerin  
HIV-1
  98.09%
Betulinic acid  
HIV-1, EC50: 1.4 μM
  98.43%
Scutellarin  
HIV-1
  98.56%
ONX-0914  
HIV-1
  99.72%
Dolutegravir  
HIV-1
  99.98%
Zidovudine  
HIV-1
  99.95%
Lopinavir  
HIV-1
  99.87%
Tenofovir  
HIV-1
  99.89%
Efavirenz  
HIV-1
  99.84%
Nelfinavir  
HIV-1
  98.83%
Raltegravir  
HIV-1
HIV-2
99.93%
3-Deazaadenosine hydrochloride  
HIV-1
  99.67%
Emtricitabine  
HIV-1
HIV-2
99.94%
Bictegravir  
HIV-1
  99.79%
Tenofovir Disoproxil fumarate  
HIV-1
  99.67%
Lenacapavir  
HIV-1
  98.48%
Nevirapine  
HIV-1
  99.93%
Stavudine  
HIV-1
HIV-2
99.87%
Cenicriviroc  
R5 HIV-1, IC50: 0.024-0.08 nM (in PBMCs)
R5 HIV-2, IC50: 0.03-0.98 nM (in PBMCs)
99.01%
TAK-779  
R5 HIV-1 (CTV), EC50: 3.5 nM (in PBMCs)
R5 HIV-1 (CTV), EC90: 27 nM (in PBMCs)
R5 HIV-1 (KK), EC50: 1.6 nM (in PBMCs)
R5 HIV-1 (KK), EC90: 20.8 nM (in PBMCs)
R5 HIV-1 (HHA), EC50: 3.2 nM (in PBMCs)
R5 HIV-1 (HHA), EC90: 7.5 nM (in PBMCs)
R5 HIV-1 (Ba-L), EC50: 1.2 nM (in MAGI-CCR5 cells)
R5 HIV-1 (Ba-L), EC50: 3.7 nM (in PBMCs)
R5 HIV-1 (Ba-L), EC90: 5.7 nM (in MAGI-CCR5 cells)
R5 HIV-1 (Ba-L), EC90: 12.8 nM (in PBMCs)
  99.73%
Limonin  
HIV-1
  98.68%
Triciribine  
HIV-1, IC50: 0.02-0.46 μM
HIV-2, IC50: 0.02-0.46 μM
99.81%
Miltefosine  
HIV-1
  ≥98.0%
Theaflavin 3,3'-digallate  
HIV-1
  99.73%
Cobicistat  
HIV-1
  99.77%
Rilpivirine  
HIV-1
  99.71%
Tenofovir alafenamide  
HIV-1
HIV-2
99.92%
Tat-beclin 1  
HIV-1
  99.68%
α-Lipoic Acid  
HIV-1
  99.86%
Indinavir sulfate  
HIV-1
  99.96%
Mavorixafor trihydrochloride  
HIV-1 (NL4.3 strain), IC50: 1 nM (in MT-4 cells)
HIV-1 (NL4.3 strain), IC50: 9 nM (in PBMCs)
HIV-1 (NL4.3 strain), IC90: 3 nM (in MT-4 cells)
HIV-1 (NL4.3 strain), IC90: 26 nM (in PBMCs)
  99.75%
5-(N,N-Hexamethylene)-amiloride  
HIV-1
  98.47%
Fangchinoline  
HIV-1
  99.92%
Elvitegravir  
HIV-1
HIV-2
BRD-K98645985  
HIV-1
  99.19%
Darunavir  
HIV-1
  99.91%
Ro24-7429  
HIV-1
  99.90%
Sennoside A  
HIV-1
  99.71%
Enfuvirtide  
HIV-1
  99.81%
Azvudine hydrochloride  
HIV-1, EC50: 0.03-6.92 nM
HIV-2, EC50: 0.018-0.02 nM
Etravirine  
HIV-1
HIV-2
99.56%
3-Deazaadenosine  
HIV-1
  99.87%
Tipranavir  
HIV-1
  ≥98.0%
Saquinavir mesylate  
HIV-1
HIV-2
99.89%
Nelfinavir Mesylate  
HIV-1
  98.93%
Tizoxanide  
HIV-1
  99.09%
Sparstolonin B  
HIV-1
  99.54%
Pentosan Polysulfate Sodium (W/W 43%)  
HIV-1
 
BRD-6929  
HIV-1
  99.04%
Temsavir  
HIV-1
  98.06%
Atazanavir sulfate  
HIV-1
  99.94%
Bromhexine hydrochloride  
HIV-1
  99.84%
IT1t dihydrochloride  
HIV-1 (X4), IC50: 14.2 nM (in MT-4 cells)
HIV-1 (X4), IC50: 19 nM (in PBMCs)
  99.77%
Tenofovir Disoproxil  
HIV-1
  99.84%
Fumagillin  
HIV-1
  ≥99.0%
PF-3450074  
HIV-1 (NL4.3 strain), IC50: 0.72 μM
  98.44%
DDX3-IN-2
HIV
    99.36%
BRD3308  
HIV-1
  98.82%
Obefazimod  
HIV-1, IC50: 0.1-0.5 μM (in PBMCs)
  99.61%
Gardiquimod diTFA  
HIV-1
  ≥99.0%
2-Hydroxyacetophenone
HIV
    99.91%
Tenofovir alafenamide fumarate  
HIV-1
HIV-2
99.14%
Cenicriviroc Mesylate  
R5 HIV-1, IC50: 0.024-0.08 nM (in PBMCs)
R5 HIV-2, IC50: 0.03-0.98 nM (in PBMCs)
99.04%
Delavirdine mesylate  
HIV-1
  99.82%
TC14012
HIV
    99.90%
Cyclotriazadisulfonamide  
HIV-1
  98.54%
Gardiquimod  
HIV-1
  99.91%
Methyl gallate  
HIV-1
  99.98%
9-Aminoacridine  
HIV-1
  99.50%
Trilobatin  
HIV-1
  99.00%
Oleanonic acid  
HIV-1
  99.63%
Atazanavir  
HIV-1
  99.86%
Fostemsavir  
HIV-1
  99.64%
L-Chicoric Acid  
HIV-1
  99.98%
Azvudine  
HIV-1, EC50: 0.03-6.92 nM
HIV-2, EC50: 0.018-0.02 nM
99.60%
2-Hydroxycinnamic acid
HIV
    98.30%
DAPTA  
HIV-1
  99.85%
Decanoyl-RVKR-CMK TFA  
HIV-1
HIV-2
99.28%
2',3'-Dideoxyadenosine  
HIV-1
HIV-2
99.89%
Bryostatin 1  
HIV-1
  99.70%
Darunavir Ethanolate  
HIV-1
  99.81%
Diphyllin  
HIV-1, IC50: 0.38 μM
  99.90%
AMD 3465 hexahydrobromide  
X4 HIV-1 (IIIB), IC50: 12.3 nM (in MT-4 cells)
X4 HIV-1 (NL4.3), IC50: 6.1 nM (in MT-4 cells)
X4 HIV-1 (NL4.3AMD3100), IC50: 2822 nM (in MT-4 cells)
X4 HIV-1 (RF), IC50: 7.4 nM (in MT-4 cells)
X4 HIV-1 (HE), IC50: 9.8 nM (in MT-4 cells)
HIV-2 (ROD), IC50: 12.3 nM (in MT-4 cells)
HIV-2 (EHO), IC50: 12.3 nM (in MT-4 cells)
≥98.0%
FC131 TFA
HIV
    99.89%
Ibalizumab  
HIV-1
  99.52%
Soyasaponin II  
HIV-1, IC50: 112 μM
  99.81%
Erythromycin Ethylsuccinate  
HIV-1
  ≥98.0%
TAT (48-57)  
HIV-1
  98.65%
Celgosivir hydrochloride  
HIV-1
  ≥98.0%
TAT peptide TFA  
HIV-1
  99.49%
PTACH  
HIV-1
  99.65%
Thiamine disulfide  
HIV-1
  98.05%
Apelin-12  
HIV-1
  99.90%
HIV-1 TAT (48-60)  
HIV-1
  99.80%
Tenofovir hydrate  
HIV-1
  ≥98.0%
Bictegravir sodium  
HIV-1
  99.71%
TAT TFA  
HIV-1
  98.40%
TAK-220  
HIV-1 (KK), EC50: 1.2 nM (in PBMCs)
HIV-1 (KK), EC90: 12 nM (in PBMCs)
HIV-1 (HNK), EC50: 1.7 nM (in PBMCs)
HIV-1 (HNK), EC90: 28 nM (in PBMCs)
HIV-1 (CTV), EC50: 0.72 nM (in PBMCs)
HIV-1 (CTV), EC90: 5 nM (in PBMCs)
HIV-1 (HKW), EC50: 1.7 nM (in PBMCs)
HIV-1 (HKW), EC90: 12 nM (in PBMCs)
HIV-1 (HHA), EC50: 0.55 nM (in PBMCs)
HIV-1 (HHA), EC90: 4 nM (in PBMCs)
HIV-1 (HTN), EC50: 0.93 nM (in PBMCs)
HIV-1 (HTN), EC90: 15 nM (in PBMCs)
  99.95%
Apelin-17(human, bovine)  
HIV-1
HIV-2
Islatravir  
HIV-1 (WT), EC50: 0.068 nM
HIV-1 (MDR), EC50: 0.15 nM
HIV-1 (M184V), EC50: 3.1 nM
  99.94%
α-Lipoic Acid-d5  
HIV-1
 
Vicriviroc maleate  
HIV-1 (JrFL), IC90: 3.3 nM (in PBMC cells)
HIV-1 (ADA-M), IC90: 2.8 nM (in PBMC cells)
HIV-1 (301657), IC90: 1.8 nM (in PBMC cells)
HIV-1 (JV1083), IC90: 4.9 nM (in PBMC cells)
HIV-1 (RU 570), IC90: 10 nM (in PBMC cells)
  99.91%
Elsulfavirine  
HIV-1
  99.63%
Apelin-36(human)  
HIV-1
HIV-2
98.11%
BMS-378806  
HIV-1
HIV-2
98.94%
NF279  
HIV-1
  ≥98.0%
HIV-1 integrase inhibitor  
HIV-1
 
LDC4297 hydrochloride  
HIV-1 (NL4.3 strain), EC50: 1.04 μM
4LIG7, EC50: 1.13 μM
  98.25%
Aplaviroc hydrochloride  
HIV-1Ba-L, IC50: 0.4 nM
HIV-1JRFL, IC50: 0.1 nM
HIV-1MOKW, IC50: 0.2 nM
  99.76%
Salicylanilide  
HIV-1
  99.90%
Chloroquine-d5  
HIV-1
  ≥99.0%
Censavudine  
HIV-1, IC50: 450-890 nM
HIV-2, EC50: 30-81 nM
98.18%
3′-Azido-2′,3′-dideoxyuridine
HIV
    99.11%
HIV-1 inhibitor-45  
HIV-1
  99.54%
Aeroplysinin 1  
HIV-1, IC50: 14.6 μM
 
Chloroquine phosphate (Standard)  
HIV-1
  99.67%
Hck-IN-1  
HIV-1 Nef, IC50: 100-300 nM
  98.53%
Tenofovir alafenamide hemifumarate  
HIV-1
HIV-2
99.70%
AMD 3465  
X4 HIV-1 (IIIB), IC50: 12.3 nM (in MT-4 cells)
X4 HIV-1 (NL4.3), IC50: 6.1 nM (in MT-4 cells)
X4 HIV-1 (NL4.3AMD3100), IC50: 2822 nM (in MT-4 cells)
X4 HIV-1 (RF), IC50: 7.4 nM (in MT-4 cells)
X4 HIV-1 (HE), IC50: 9.8 nM (in MT-4 cells)
HIV-2 (ROD), IC50: 12.3 nM (in MT-4 cells)
HIV-2 (EHO), IC50: 12.3 nM (in MT-4 cells)
99.59%
Fostemsavir Tris  
HIV-1
  99.94%
Rovafovir etalafenamide  
HIV-1
HIV-2
FGI-106 tetrahydrochloride  
HIV-1
  99.68%
Fipravirimat dihydrochloride  
HIV-1
 
Tenofovir exalidex  
HIV-1
HIV-2
98.70%
Ulonivirine  
HIV-1
  98.31%
Nifeviroc  
HIV-1
  98.17%
Ingenol-3-palmitate  
HIV-1, IC50: 4.1 nM
  99.54%
FNC-TP  
HIV-1
  99.92%
Claficapavir  
HIV-1
  99.14%
α-Lipoic Acid (Standard)  
HIV-1
  99.90%
Zingibroside R1  
HIV-1
  99.75%
Azulene
HIV
    99.98%
Kaempferol-3-O-(6′′-galloyl)-β-glucopyranoside    
HIV-2
99.26%
Formycin A  
HIV-1, EC50: 10 μM
  ≥99.0%
3'-Azido-3'-deoxy-5-methylcytidine  
HIV-1, EC50: 0.06 μM (in PBM cells)
  99.15%
SARS-CoV-IN-3  
HIV-1
  99.36%
Fipravirimat  
HIV-1
 
Celgosivir  
HIV-1
 
SARS-CoV-IN-2  
HIV-1
  98.66%
HIV-1 inhibitor-8  
HIV-1 (WT), IC50: 0.081 μM
  98.03%
Reverse transcriptase-IN-1  
HIV-1
  98.08%
IT1t  
HIV-1 (X4), IC50: 14.2 nM (in MT-4 cells)
HIV-1 (X4), IC50: 19 nM (in PBMCs)
 
DPC-681  
HIV-1
  99.89%
Apelin-36(human) TFA  
HIV-1
HIV-2
98.11%
Doxorubicin  
HIV-1
 
Gomisin M2
HIV, EC50: 2.4 μM
    99.87%
Aplaviroc  
HIV-1Ba-L, IC50: 0.4 nM
HIV-1JRFL, IC50: 0.1 nM
HIV-1MOKW, IC50: 0.2 nM
 
HIV-1 inhibitor-6  
X4 HIV-1 (IIIB), EC50: 0.6 μM
R5 HIV-1, EC50: 0.9 μM
  98.91%
FNC-TP trisodium  
HIV-1
 
AzddMeC  
HIV-1, EC50: 9 nM (Human PBM cells)
HIV-1, EC50: 6 nM (Human macrophages)
  98.96%
EFdA-TP tetraammonium  
HIV-1
  98.03%
EFdA-TP tetrasodium  
HIV-1
 
Pentosan Polysulfate  
HIV-1
 
Gomisin M1  
HIV-1
  99.56%
Suvizumab  
HIV-189.6, IC50: 0.2 μg/mL
HIV-1MN, IC50: 0.1 μg/mL
HIV-1SF2, IC50: 1.0 μg/mL
 
Mavorixafor  
HIV-1 (NL4.3 strain), IC50: 1 nM (in MT-4 cells)
HIV-1 (NL4.3 strain), IC50: 9 nM (in PBMCs)
HIV-1 (NL4.3 strain), IC90: 3 nM (in MT-4 cells)
HIV-1 (NL4.3 strain), IC90: 26 nM (in PBMCs)
 
KRH-3955 hydrochloride  
X4 HIV-1NL4-3, EC50: 0.3-1.0 nM
 
Apelin-36(rat, mouse)  
HIV-1
HIV-2
98.07%
FC131
HIV
   
NBD-557  
HIV-1
  99.41%
9-Propenyladenine  
HIV-1
 
Indinavir  
HIV-1
 
Dolutegravir intermediate-1  
HIV-1
  99.80%
(Z)-9-Propenyladenine  
HIV-1
  98.02%
Chloroquine dihydrochloride  
HIV-1
 
Panobinostat lactate  
HIV-1
 
Mavorixafor hydrochloride  
HIV-1 (NL4.3 strain), IC50: 1 nM (In MT-4 cells)
HIV-1 (NL4.3 strain), IC50: 9 nM (In PBMCs)
HIV-1 (NL4.3 strain), IC90: 3 nM (In MT-4 cells)
HIV-1 (NL4.3 strain), IC90: 26 nM (In PBMCs)
 
NBD-14270  
HIV-1
  98.47%
FGI-106  
HIV-1
 
NBD-14189  
HIV-1
  99.84%
HIV-1 inhibitor-33  
HIV-1 (WT), EC50: 8.6 nM
 
HIV-1 inhibitor-51  
HIV-1 (WT), IC50: 0.03 μM
HIV-1 (WT), Kd: 2.5 μM
HIV-1 (L100I), EC50: 3.04 nM
HIV-1 (K103N), EC50: 2.87 nM
HIV-1 (Y181C), EC50: 10.2 nM
HIV-1 (Y188L), EC50: 13.2 nM
HIV-1 (E138K), EC50: 9.77 nM
HIV-1 (F227L+V106A), EC50: 19.8 nM
HIV-1 (RES056), EC50: 53.3 nM
 
Wikstrol A  
HIV-1, IC50: 67.8
 
HIV-1 inhibitor-16  
HIV-1 (WT), EC50: 1.3 nM
HIV-1 (K103N), EC50: 5.4 nM
HIV-1 (E138K), EC50: 9.2 nM
HIV-1 (Y181C), EC50: 22 nM
HIV-1 (L100I), EC50: 35 mM
 
Siamycin I  
HIV-1
HIV-2
CCR5 antagonist 3  
HIV-1, EC50: 0.010 μM (In TZM-bl cells)
 
HIV-1 inhibitor-44  
HIV-1, EC50: 0.209 μM
 
HIV-1 Nef-IN-1  
HIV-1 Nef, Kd: 6.7 μM
  98.60%
Kadsuracoccinic acid A  
HIV-1, EC50: 68.7 μM
 
INCB9471  
HIV-1
 
Fuscin
HIV
   
H-Gly-Pro-Gly-NH2  
HIV (IIIB), EC50: 35 μM
HIV-2 (ROD), EC50: 30 μM
BMS 561390  
HIV-1 (WT), IC50: 2.0 nM
HIV-1 (K103N), IC50: 21 nM
HIV-1 (L100I), IC50: 5.9 nM
 
HIV-1 inhibitor-34  
HIV-1 (WT), EC50: 6.4 nM
 
Fosdevirine  
HIV-1 (K103N)
HIV-1 (Y181C)
HIV-1
 
HIV-1 Rev (34-50)  
HIV-1
 
PROTAC Vif degrader-1  
HIV (IIIB), EC50: 33.35 μM
 
Reverse transcriptase-IN-3  
HIV (IIIB), EC50: 8 nM
HIV-1 (L100I), EC50: 65 nM
HIV-1 (K103N), EC50: 9 nM
HIV-1 (Y181C), EC50: 45 nM
HIV-1 (Y188L), EC50: 35 nM
HIV-1 (E138K), EC50: 0.734 μM
HIV-1 (F227L+V106A), EC50: 34 nM
HIV-1 (RES056), EC50: 42 nM
 
IQP-0528  
HIV-1
HIV-2
99.90%
Luzopeptin A  
HIV-1 RT, IC50: 7 nM
HIV-2 RT, IC50: 68 nM
Inophyllum B  
HIV-1, IC50: 1.4 μM
 
Corydine  
HIV-1
 
Nevirapine-d4  
HIV-1
 
HIV-1 inhibitor-29  
HIV (IIIB), EC50: 2.18 μM
HIV-1 (F227L/V106A), EC50: 0.974 μM
 
WRNA10
HIV, IC50: 10 μM (CC50: 40 μM[1])
   
Sennoside A (Standard)  
HIV-1
 
HIV-1 inhibitor-64  
HIV-1 (WT)
 
HIV-1 inhibitor-40  
HIV-1 (WT), EC50: 1.9 nM
HIV-1 (L100I), EC50: 0.019 μM
HIV-1 (K103N), EC50: 0.004 μM
HIV-1 (Y181C), EC50: 0.029 μM
HIV-1 (Y188L), EC50: 0.570 μM
HIV-1 (E138K), EC50: 0.009 μM
 
4'-Ethynyl-2'-deoxyadenosine  
HIV-1
 
TC14012 TFA
HIV
   
AIC-292  
HIV-1
 
HIV-IN-5  
HIV-1, IC50: 0.16 ± 0.0 μM
HIV-1 (Y181C), IC50: >100 μM
HIV-1 (K103N), IC50: >100 μM
 
HIV-1 inhibitor-13  
HIV-1 (WT), EC50: 2.85 ± 1.1 nM
 
HIV-1 inhibitor-15  
HIV-1 (WT), EC50: 1.7 nM
HIV-1 (L100I), EC50: 4 nM
HIV-1 (K103N), EC50: 2 nM
HIV-1 (Y181C), EC50: 6 nM
HIV-1 (E138K), EC50: 9 nM
 
Patentiflorin A  
HIV-1
 
HIV-1 inhibitor-46  
HIV-1, EC50: 1.425 μM
 
HIV-1 inhibitor-39  
HIV-1, EC50: >112.88 μM
 
Emtricitabine S-oxide
HIV
   
HIV-1 inhibitor-30  
HIV-1 (WT), EC50: 40 nM
RT-K103N, EC50: 0.72 μM
RT-Y181C, EC50: 0.04 μM
RT-K103N,Y181C, EC50: 0.69 μM
RT-L100I,K103N, EC50: 0.43 μM
RT-Y188L, EC50: 1.42 μM
RT-K103N,G190A, EC50: 0.70 μM
RT-K103N,V108I, EC50: 0.56 μM
 
HIV-1 inhibitor-22  
HIV-1 (WT), EC50: 0.304 μM
HIV-1 (K103N), EC50: 0.201 μM
 
Myriceric acid B  
HIV-1, IC50: 8.3±0.2 μg/mL (infection of HIV-1 Env pseudovirus)
 
Dexelvucitabine  
HIV-1
  99.52%
CCR5 antagonist 2  
HIV-1, EC50: 11 nM (TZM-bl cell)
 
Apelin-36(rat, mouse) TFA  
HIV-1
HIV-2
HIV-1 inhibitor-28  
HIV-1 (WT), EC50: 58 nM
 
AL-470  
HIV-1, EC50: 0.27 μM
HIV-2, EC50: 0.63 μM
CCR5 antagonist 1
HIV
   
HIV-1 inhibitor-24  
HIV-1 (WT), EC50: 1.6 nM
 
Peptide T TFA  
HIV-1
 
HIV-1 inhibitor-54  
HIV-1
 
HIV-1 inhibitor-21  
HIV-1 (WT), EC50: 12.7 nM
HIV-1 (K103N), EC50: 10.4 nM
 
HIV-1 inhibitor-25  
HIV (IIIB), EC50: 13.6 nM
HIV-1 (L100I), EC50: 1.2458 ± 0 μM
HIV-1 (K103N), EC50: 0.4383 ± 0 μM
HIV-1 (Y181C), EC50: 0.5075 ± 0 μM
HIV-1 (Y188L), EC50: 5.8136 ± 2 μM
HIV-1 (E138K), EC50: 0.1961 ± 0 μM
HIV-1 (F227L+V106A), EC50: 3.0683 ± 0 μM
 
HIV-1 protease-IN-6  
HIV-1
 
CXCR4 antagonist 4
HIV, IC50: 7 nM
   
Calcium mesoxalate  
HIV-1
 
CI-39  
HIV-1 (WT), EC50: 3.40 μM
HIV-1 (WT), CC50: >30 μM
 
HIV-1 inhibitor-32  
HIV-1 (WT), IC50: 34 nM
 
Atazanavir-d15  
HIV-1
 
HIV-1 protease-IN-4  
HIV-1
 
HIV-1 inhibitor-52  
HIV-1 (WT), EC50: 1.6 nM
HIV-1 V370A, EC50: 3.0 nM
HIV-1 ΔV370, EC50: 5.1 nM
HIV-1 V362I/V370A, EC50: 2.0 nM
HIV-1 T332S/V362I/prR41G, EC50: 6.4 nM
HIV-1 A326T/V362I/V370A, EC50: 4.3 nM
HIV-1 R361K/V362I/L363M, EC50: 4.5 nM
 
HIV-1 inhibitor-18  
HIV-1 NL4-3, EC50: 5.14 μM
 
HIV-1 inhibitor-14  
HIV-1 (WT), EC50: 6.17 nM
HIV-1 (L100I), EC50: 12.4 nM
HIV-1 (K103N), EC50: 6.91 nM
HIV-1 (Y181C), EC50: 8.91 nM
HIV-1 (Y188L), EC50: 7.66 nM
HIV-1 (F227L+V106A), EC50: 5.79 nM
HIV-1 (K103N+Y181C), EC50: 27.9 nM
HIV-1 (E138K), EC50: 7.66 nM
 
gp120-IN-2  
HIV-1, IC50: 7.5 μM
HIV-1, CC50: 112.93 μM
 
HIV-1 inhibitor-23  
HIV-1 (WT), EC50: 24.9 nM
HIV-1 (K103N), EC50: 10.4 nM
 
Apelin-17(human, bovine) TFA  
HIV-1
HIV-2
DMJ-I-228  
HIV-1
 
Azt-pmap  
HIV-1
 
HIV-1 inhibitor-27  
HIV-1 YU2, IC50: 16 μM
HIV-1 NL4-3, IC50: 0.5 μM
HIV-1 89.6, IC50: 0.39 μM
 
HIV-1 inhibitor-49  
HIV-1 (WT), EC50: 17 nM
HIV-1 (L100I), EC50: 0.38 μM
HIV-1 (K103N), EC50: 2.64 μM
HIV-1 (Y181C), EC50: 1.85 μM
HIV-1 (E138K), EC50: 0.09 μM
 
SAMT-247  
HIV-1IIIB, EC50: 0.6 μM
 
CXCR4 antagonist 1  
HIV-1
 
EFdA-TP  
HIV-1
 
[(Cys(Bzl)84,Glu(OBzl)85)]CD4 (81-92)  
HIV-1
 
gp120-IN-1  
HIV-1, IC50: 2.2 μM
HIV-1, CC50: 100.90 μM
 
α-Lipoic Acid sodium  
HIV-1
 
Cys-TAT(47-57)  
HIV-1
 
DENV-IN-6  
HIV (IIIB)
 
Fozivudine tidoxil
HIV
   
HIV-1 inhibitor-43  
HIV-1 (Y188L), EC50: 21.3 nM
HIV-1 (K103N+Y181C), EC50: 6.2 nM
HIV-1 (K103N), EC50: <0.7 nM
HIV-1 (Y181C), EC50: <0.7 nM
 
Apricitabine  
HIV-1
 
Leptomycin A  
HIV-1
  ≥99.0%
DENV-IN-5  
HIV (IIIB), EC50: 0.1512 μM
 
ZLM-66  
HIV-1 (WT), EC50: 13 nM
HIV-1 (K103N), EC50: 13 nM
HIV-1 (L100I), EC50: 24 nM
HIV-1 (E138K), EC50: 25 nM
HIV-1 (Y181C), EC50: 58 nM
HIV-1 (K103N+Y181C), EC50: 260 nM
HIV-1 (F227L+V106A), EC50: 27530 nM
 
ICeD-2  
HIV-1
 
HIV-1 inhibitor-41  
HIV-1 (WT), IC50: 20.8 nM
HIV-1 (E138K), IC50: 50 nM
HIV-1 (L100I), IC50: 1.03 μM
HIV-1 (K103N), IC50: 3.39 μM
HIV-1 (Y181C), IC50: 0.75 μM
HIV-1 (Y188L), IC50: 69.04 μM
 
UC-781  
HIV-1, IC50: 0.005 μM
 
HIV-1 capsid inhibitor 1  
HIV-1, EC50: 3.13 μM
 
12-Oxocalanolide A  
HIV-1
 
HF50731  
HIV-1, IC50: 1.5 μM
 
Clavirolide L  
HIV-1
 
HIV-1 inhibitor-17  
HIV-1 NL4-3, EC50: 2.57 μM
 
HIV-1 inhibitor-12  
HIV-1
 
MIV-150  
HIV-1, EC50: <1 nM
HIV-2, EC50: <1 nM
Atazanavir-d18  
HIV-1
 
Tat-beclin 1 TFA  
HIV-1
HIV-1
 
MPG, HIV related  
HIV-1
 
Indinavir sulfate ethanolate  
HIV-1
 
Aureothin
HIV, IC50: 5.3 nM
   
HIV-1 inhibitor-42  
HIV-1, IC50: 0.06 ± 0.0 μM
HIV-1 (Y181C), IC50: 15.510 ± 1 μM
HIV-1 (K103N), IC50: 53.045 ± 6 μM
 
Efavirenz-13C6  
HIV-1
 
Scirpusin A  
HIV-1, EC50: 7 μg/mL
 
BMS-585248  
HIV-1
 
TAT (48-57) (TFA)  
HIV-1
 
HIV-1 inhibitor-50  
HIV-1 (WT), EC50: 3.04 nM
HIV-1 (L100I), EC50: 3.04 nM
HIV-1 (K103N), EC50: 2.87 nM
HIV-1 (Y181C), EC50: 10.2 nM
HIV-1 (Y188L), EC50: 13.2 nM
HIV-1 (E138K), EC50: 9.77 nM
HIV-1 (F227L+V106A), EC50: 19.8 nM
 
Crotoniazide  
HIV-1, EC50: 11 μg/mL
HIV-2 (ROD), EC50: 11 μg/mL
Stavudine sodium  
HIV-1
HIV-2
beta-L-D4A  
HIV-1
 
HIV-1 inhibitor-63  
HIV-1
 
Tenofovir maleate  
HIV-1
 
SDZ283-910  
HIV-1
 
Hinnuliquinone  
HIV-1
 
7-Deaza-2',3'-dideoxyguanosine  
HIV-1
  98.02%
TAT  
HIV-1