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Imidazo[1,2,4] triazole derivatives

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6038

Inhibitors & Agonists

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444

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491

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1593

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Products

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Targets Recommended: Amino Acid Derivatives Drug Derivative

Cat. No.	Product Name	Target	Research Areas	Chemical Structure

HY-Y0219

1,2,4-Triazole s-triazole; Pyrrodiazole	Biochemical Assay Reagents	Others
1,2,4-Triazole is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-Y0219A

*1,2,4-Triazole* sodium** s-triazole sodium; Pyrrodiazole sodium	Biochemical Assay Reagents	Infection
1,2,4-Triazole (sodium) is a biochemical reagent that can be used as a biological material or organic compound for life science related research .

HY-Y0219R

*1,2,4-Triazole* (Standard)**	Biochemical Assay Reagents	Others
1,2,4-Triazole (Standard) is the analytical standard of 1,2,4-Triazole. This product is intended for research and analytical applications. 1,2,4-Triazole is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-W113615

4-Phenyl-1H-1,2,3-triazole	Indoleamine 2,3-Dioxygenase (IDO)	Cancer
4-Phenyl-1H-1,2,3-triazole is an IDO1 inhibitor (IC₅₀: 60 μM). 4-Phenyl-1H-1,2,3-triazole can be used for cancer research .

HY-107870

*1,2,4-Triazole-3-carboxylic acid, 97%*	Biochemical Assay Reagents	Others
1,2,4-Triazole-3-carboxylic acid, 97% is a biochemical assay reagent.

HY-W012991

3-Mercapto-1,2,4-triazole	Biochemical Assay Reagents	Others
1,2-Dihydro-3H-1,2,4-triazole-3-thione is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-141652

N-2-Azidoethyl betulonamide	Drug Intermediate	Cancer
N-2-Azidoethyl betulonamide is the building block, that could generate cytotoxic triazole derivative through click chemistry .

HY-76802

Calcitriol Derivatives	VD/VDR	Metabolic Disease
Calcitriol Derivatives is a vitamin D3 analog.

HY-169368

*Thalidomide-O-Triazole-C4-amino*	E3 Ligase Ligand-Linker Conjugates	Cancer
Thalidomide-O-Triazole-C4-amino is an E3 ligase ligand-linker conjugate. Thalidomide-O-Triazole-C4-amino can be used to synthesize aTAG 4531 (HY-163168) .

HY-163107

Antimycobacterial agent-7	Bacterial	Infection
Antimycobacterial agent-7 (compound 4) is a 1,2,4-triazole anti-tuberculosis agent (MIC: 2 μg/mL). Antimycobacterial agent-7 inhibits Mtb KatG and causes the accumulation of ROS in Mtb cells. ROS produces oxidative damage, leading to the death of Mtb .

HY-141941S

Triazole Lactic Acid-13C2, 15N3	Isotope-Labeled Compounds	Others
Triazole Lactic Acid- ¹³C₂, ¹⁵N₃ is the ¹³C and ¹⁵N labeled Triazole Lactic Acid[1].

HY-100284

*Thiazolidinone-Derivatives-1*	Drug Derivative	Inflammation/Immunology
Thiazolidinone-Derivatives-1 is an antiulcer agent which inhibits the secretion of gastric acid.

HY-W331786

Ipconazole	Bacterial	Infection
Ipconazole is a triazole fungicide that can be used for treating rice seed .

HY-W007685

*Methyl 1H-1,2,4-triazole-5-carboxylate*	Biochemical Assay Reagents	Others
Methyl 1H-1,2,4-triazole-3-carboxylate is a biochemical reagent that can be used as a biological material or organic compound for life science related research.

HY-163789

*Desthiobiotin-PEG3-triazole-DBCO-sulfo-Maleimide*	ADC Linker	Cancer
Desthiobiotin-PEG3-triazole-DBCO-sulfo-Maleimide is an ADC linker used in the synthesis of antibody-drug conjugates (ADCs). Desthiobiotin-PEG3-triazole-DBCO-sulfo-Maleimide is a click chemistry reagent, it contains a DBCO group that can undergo strain-promoted alkyne-azide cycloaddition (SPAAC) with molecules containing Azide groups .

HY-W586475

*Fluorescein-triazole-PEG5-DOTA*	Radionuclide-Drug Conjugates (RDCs)	Cancer
Fluorescein-triazole-PEG5-DOTA is a radionuclide conjugate (RDC), which is capable of binding to a radionuclide. RDC has the ability to specifically target biomolecules and can be used in medical imaging or therapy .

HY-46369

*1-p-Chlorobenzyl-1,2,3-triazole-5′-O-DMT-dU Phosphoramidite*	DNA/RNA Synthesis	Others
1-p-Chlorobenzyl-1,2,3-triazole-5′-O-DMT-dU Phosphoramidite is a phosphorite monomer that can be used in the synthesis of oligonucleotides.

HY-W098127S

*Methyl 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxylate-d2*	Isotope-Labeled Compounds	Others
Methyl 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxylate-d₂ is the deuterium labeled Methyl 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxylate[1].

HY-W331786R

Ipconazole (Standard)	Bacterial	Infection
Ipconazole (Standard) is the analytical standard of Ipconazole. This product is intended for research and analytical applications. Ipconazole is a triazole fungicide that can be used for treating rice seed .

HY-168006

NSC819701	p97 ATP Synthase	Cancer
NSC819701 is a triazole inhibitor of the p97 ATPase. NSC819701 inhibits the activity of p97 ATPase by binding to a specific site of p97 .

HY-W019852

Flutriafol	Fungal	Infection
Flutriafol is a triazole fungicide with broad spectrum fungicidal activity.

HY-B2058

Triticonazole	Fungal	Infection
Triticonazole is a triazole pesticide. Triticonazole is an azole fungicide and shows endocrine disrupting activities .

HY-168005

NSC799462	p97 ATP Synthase	Cancer
NSC799462 is a triazole inhibitor of p97 ATPase. NSC799462 inhibits p97 ATPase activity (IC₅₀ = 15 nM) by binding to a specific site on p97 and causing local changes in the p97 structure .

HY-W019852R

Flutriafol (Standard)	Fungal	Infection
Flutriafol (Standard) is the analytical standard of Flutriafol. This product is intended for research and analytical applications. Flutriafol is a triazole fungicide with broad spectrum fungicidal activity.

HY-144426

Neuraminidase-IN-6	Influenza Virus	Infection
Neuraminidase-IN-6 (Compound 5c) is a potent inhibitor of neuraminidase with an IC₅₀ of 0.11 μM. Neuraminidase-IN-6 is a 1,3,4-triazole-3-acetamide derivative. Neuraminidase (NA) is an ideal target for the development of anti-influenza agents .

HY-B0847

Propiconazole 1 Publications Verification	Fungal Reactive Oxygen Species	Infection
Propiconazole is an orally active N-substituted triazole used as a fungicide. Propiconazole is a mouse liver hepatotoxicant and a hepatocarcinogen that has adverse reproductive and developmental toxicities in experimental animals .

HY-B2058R

Triticonazole (Standard)	Fungal	Infection
Triticonazole (Standard) is the analytical standard of Triticonazole. This product is intended for research and analytical applications. Triticonazole is a triazole pesticide. Triticonazole is an azole fungicide and shows endocrine disrupting activities .

HY-126677

*Boc-NH-PEG3-C2-triazole-DBCO-PEG4-VC-PAB-DMEA*	ADC Linker PROTAC Linkers	Cancer
Boc-NH-PEG3-C2-triazole-DBCO-PEG4-VC-PAB-DMEA is a double claevable 3-unit and 4-unit PEG linker for antibody-agent-conjugation (ADC). Boc-NH-PEG3-C2-triazole-DBCO-PEG4-VC-PAB-DMEA also is a PROTAC linker that can be used in the synthesis of PROTACs.

HY-B0847R

Propiconazole (Standard)	Fungal Reactive Oxygen Species	Infection
Propiconazole (Standard) is the analytical standard of Propiconazole. This product is intended for research and analytical applications. Propiconazole is an orally active N-substituted triazole used as a fungicide. Propiconazole is a mouse liver hepatotoxicant and a hepatocarcinogen that has adverse reproductive and developmental toxicities in experimental animals .

HY-14273S

Isavuconazole-d4 BAL-4815-d₄; RO-0094815-d₄	Fungal Cytochrome P450	Infection
Isavuconazole-d₄ is a deuterium labeled Isavuconazole (BAL-4815). Isavuconazole is a triazole proagent with antifungal activity against yeasts, molds, and dimorphic fungi[1].

HY-157532

AChE-IN-55	Cholinesterase (ChE)	Others
AChE-IN-55, 1,2,3-Triazole oxime derivative, is an inhibitor of AChE(4.8 μM) .

HY-76200

Voriconazole 5+ Cited Publications UK-109496	Fungal Bacterial	Infection Cancer
Voriconazole (UK-109496) is a second-generation, broad-spectrum triazole antifungal agent that inhibits fungal ergosterol biosynthesis. Voriconazole exerts its antifungal activity by inhibition of 14-α-lanosterol demethylation, which is mediated by fungal cytochrome P450 enzymes .

HY-76200B

Voriconazole camphorsulfonate UK-109496 camphorsulfonate	Fungal Bacterial	Infection Cancer
Voriconazole (UK-109496) camphorsulfonate is a second-generation, broad-spectrum triazole antifungal agent that inhibits fungal ergosterol biosynthesis. Voriconazole camphorsulfonate exerts its antifungal activity by inhibition of 14-α-lanosterol demethylation, which is mediated by fungal cytochrome P450 enzymes .

HY-14273

Isavuconazole 4 Publications Verification BAL-4815; RO-0094815	Fungal Cytochrome P450 Antibiotic	Infection Cancer
Isavuconazole (BAL-4815) is a triazole proagent with antifungal activity against yeasts, molds, and dimorphic fungi. Isavuconazole inhibits ergosterol biosynthesis and results in the disruption of fungal membrane structure and function. Isavuconazole is a moderate inhibitor of CYP3A4.

HY-14273R

Isavuconazole (Standard)	Fungal Cytochrome P450 Antibiotic	Infection
Isavuconazole (Standard) is the analytical standard of Isavuconazole. This product is intended for research and analytical applications. Isavuconazole (BAL-4815) is a triazole proagent with antifungal activity against yeasts, molds, and dimorphic fungi. Isavuconazole inhibits ergosterol biosynthesis and results in the disruption of fungal membrane structure and function. Isavuconazole is a moderate inhibitor of CYP3A4.

HY-161812

MOR agonist-4	Opioid Receptor	Others
MOR agonist-4 (2d) is a G protein signaling-biased Kappa opioid receptor (KOR) agonist with an EC₅₀ value of 11 nM. MOR agonist-4 contains an electron withdrawing CF3 group and a bias factor of 38 based on triazole. MOR agonist-4 is used in the research of pruritis and analgesia .

HY-117766

PC945	Fungal Cytochrome P450	Infection
PC945, a potent, long-acting antifungal triazole, possesses activity against a broad range of both azole-susceptible and azole-resistant strains of Aspergillus fumigatus. PC945 is also a potent, tightly binding inhibitor of A. fumigatus sterol 14α-demethylase activity, CYP51A and CYP51B, with IC₅₀s of 0.23 μM and 0.22 μM, respectively .

HY-B0101

Fluconazole 10+ Cited Publications UK-49858	Fungal Antibiotic Bacterial	Infection Cancer
Fluconazole (UK-49858) is a triazole antifungal agent with excellent activities against a broad range of fungi, especially against Candida albicans. Fluconazole inhibits C. albicans and Candida kefyr with IC₉₉s range from 0.20 μg/mL to 0.39 μg/mL .

HY-16506

Trimethaphan camsylate Ro 2-2222; Thiophanium derivatives	Adrenergic Receptor	Cardiovascular Disease Others
Trimethaphan camsylate is an arterial blood pressure lowering agent that has been shown to reduce pulmonary venous pressure in experimental pulmonary edema.

HY-17514

Itraconazole 15+ Cited Publications R51211	Fungal Hedgehog Cytochrome P450 Autophagy Antibiotic Bacterial	Infection Cancer
Itraconazole (R51211) is a triazole antifungal agent and a potent and orally active Hedgehog (Hh) signaling pathway antagonist with an IC₅₀ of ~800 nM. Itraconazole potently inhibits lanosterol 14α-demethylase (cytochrome P450 enzyme), thereby inhibits the oxidative conversion of lanosterol to ergosterol. Itraconazole has anticancer and antiangiogenic effects. Itraconazole is a oxysterol-binding protein (OSBP) inhibitor .

HY-B0101R

Fluconazole (Standard)	Fungal Antibiotic Bacterial	Infection Cancer
Fluconazole (Standard) is the analytical standard of Fluconazole. This product is intended for research and analytical applications. Fluconazole (UK-49858) is a triazole antifungal agent with excellent activities against a broad range of fungi, especially against Candida albicans. Fluconazole inhibits C. albicans and Candida kefyr with IC99s range from 0.20 μg/mL to 0.39 μg/mL .

HY-172001

α-GalCer analog 8	Drug Derivative	Cancer
α-GalCer analog 8 is a triazole derivative of α-Galactosylceramide (HY-102022). α-Galactosylceramide is a synthetic glycolipid with antitumorial and immunostimulatory .

HY-P10472

Azaline B	GnRH Receptor	Endocrinology
Azaline B is an antagonist for gonadotropin-releasing hormone (GnRH) with IC₅₀ of 1.37 nM, Azaline B can be used in research of sex hormone-related pathological states, ovulation induction and male contraception .

HY-17514R

Itraconazole (Standard)	Fungal Hedgehog Cytochrome P450 Autophagy Antibiotic Bacterial	Infection Cancer
Itraconazole (Standard) is the analytical standard of Itraconazole. This product is intended for research and analytical applications. Itraconazole (R51211) is a triazole antifungal agent and a potent and orally active Hedgehog (Hh) signaling pathway antagonist with an IC50 of ~800 nM. Itraconazole potently inhibits lanosterol 14α-demethylase (cytochrome P450 enzyme), thereby inhibits the oxidative conversion of lanosterol to ergosterol. Itraconazole has anticancer and antiangiogenic effects. Itraconazole is a oxysterol-binding protein (OSBP) inhibitor .

HY-W291634

H-D-Glu-OtBu hydrochloride	Amino Acid Derivatives	Others
H-D-Glu-OtBu (hydrochloride) is a glutamic acid derivative .

HY-41912B

Boc-D-norleucine Boc-D-Nle-OH; N-BOC-D-norleucine	Amino Acid Derivatives	Others
Boc-D-norleucine (Boc-D-Nle-OH) is a leucine derivative that can be used for peptide synthesis .

HY-W013726

Fmoc-Phe(4-Br)-OH	Amino Acid Derivatives	Others
Fmoc-Phe(4-Br)-OH is a phenylalanine derivative that can be used for compound synthesis .

HY-W033132

N-(2-Methoxyethyl)-N-methylglycine	Amino Acid Derivatives	Others
N-(2-Methoxyethyl)-N-methylglycine is a glycine derivative that can be used for compound synthesis .

HY-W007052

Fmoc-alpha-allyl-L-alanine Fmoc-(Me)Gly(Allyl)-OH	Amino Acid Derivatives	Others
Fmoc-alpha-allyl-L-alanine is an Fmoc-protected alanine derivative.

HY-W013152

Fmoc-Phe(3-Me)-OH	Amino Acid Derivatives	Others
Fmoc-Phe(3-Me)-OH is a Fmoc-protected phenylalanine derivative .

Cat. No.	Product Name	Category	Target	Chemical Structure

HY-76200

Voriconazole 5+ Cited Publications UK-109496	Microorganisms Source classification	Fungal Bacterial
Voriconazole (UK-109496) is a second-generation, broad-spectrum triazole antifungal agent that inhibits fungal ergosterol biosynthesis. Voriconazole exerts its antifungal activity by inhibition of 14-α-lanosterol demethylation, which is mediated by fungal cytochrome P450 enzymes .

HY-B0101

Fluconazole 10+ Cited Publications UK-49858	Microorganisms Source classification	Fungal Antibiotic Bacterial
Fluconazole (UK-49858) is a triazole antifungal agent with excellent activities against a broad range of fungi, especially against Candida albicans. Fluconazole inhibits C. albicans and Candida kefyr with IC₉₉s range from 0.20 μg/mL to 0.39 μg/mL .

HY-17514

Itraconazole 15+ Cited Publications R51211	Microorganisms Source classification	Fungal Hedgehog Cytochrome P450 Autophagy Antibiotic Bacterial
Itraconazole (R51211) is a triazole antifungal agent and a potent and orally active Hedgehog (Hh) signaling pathway antagonist with an IC₅₀ of ~800 nM. Itraconazole potently inhibits lanosterol 14α-demethylase (cytochrome P450 enzyme), thereby inhibits the oxidative conversion of lanosterol to ergosterol. Itraconazole has anticancer and antiangiogenic effects. Itraconazole is a oxysterol-binding protein (OSBP) inhibitor .

HY-N1977

Podophyllotoxin glucoside	other families Classification of Application Fields Source classification Lignans Phenylpropanoids Plants Disease Research Fields Cancer	Others
Podophyllotoxin glucoside is a podophyllotoxin derivative, has anti-tumor effects .

HY-20897A

5-Bromo-L-tryptophan	Structural Classification Natural Products Classification of Application Fields Source classification Other Diseases Endogenous metabolite Disease Research Fields	Endogenous Metabolite
5-Bromo-L-tryptophan is an α-amino acid derivative that can be found in Semenospongia sp. .

HY-B0101R

Fluconazole (Standard)	Microorganisms Source classification	Fungal Antibiotic Bacterial
Fluconazole (Standard) is the analytical standard of Fluconazole. This product is intended for research and analytical applications. Fluconazole (UK-49858) is a triazole antifungal agent with excellent activities against a broad range of fungi, especially against Candida albicans. Fluconazole inhibits C. albicans and Candida kefyr with IC99s range from 0.20 μg/mL to 0.39 μg/mL .

HY-17514R

Itraconazole (Standard)	Microorganisms Source classification	Fungal Hedgehog Cytochrome P450 Autophagy Antibiotic Bacterial
Itraconazole (Standard) is the analytical standard of Itraconazole. This product is intended for research and analytical applications. Itraconazole (R51211) is a triazole antifungal agent and a potent and orally active Hedgehog (Hh) signaling pathway antagonist with an IC50 of ~800 nM. Itraconazole potently inhibits lanosterol 14α-demethylase (cytochrome P450 enzyme), thereby inhibits the oxidative conversion of lanosterol to ergosterol. Itraconazole has anticancer and antiangiogenic effects. Itraconazole is a oxysterol-binding protein (OSBP) inhibitor .

HY-N11966

2'-Hydroxylagarotetrol	Structural Classification Monophenols Thymelaeaceae Source classification Phenols Plants Aquilaria sinensis (Lour.) Spreng.	Others
2'-Hydroxylagarotetrol is a phenylethychromone derivative .

HY-N8791

Qianhucoumarin G	Structural Classification Chrysanthemum × morifolium (Ramat.) Hemsl. Source classification Coumarins Phenylpropanoids Plants Umbelliferae	Others
Qianhucoumarin G is a natural coumarin derivative found in Ligustici Radix .

HY-N11974

Isobatatasin I	Structural Classification Monophenols Tamus communis L. Source classification Phenols Plants Dioscoreaceae	Others
Isobatatasin I is a phenanthrene derivative that can be isolated from the rhizome of safflower .

HY-N0947

(-)-Anomalin (-)-Praeruptorin B	Structural Classification Classification of Application Fields Source classification Coumarins Salvia hypargeia Fisch. & C.A.Mey. Phenylpropanoids Umbelliferae Plants Inflammation/Immunology Disease Research Fields Artemisia vulgaris L.	Others
(-)-Anomalin ((-)-Praeruptorin B) is a coumarin derivative isolated from the root of Angelica anomala .

HY-N15447

Visnaginone	Thymus serpyllum L. Structural Classification Natural Products Source classification Umbelliferae Plants	Drug Derivative
Visnaginone is the derivative of Visnagin (HY-N1082). Visnagin, an antioxidant furanocoumarin derivative, possess anti-inflammatory and analgesic properties. Visnagin has substantial potential to prevent Cerulein induced acute pancreatitis (AP). Visnagin possess promising vasodilator effects in vascular smooth muscles .

HY-116189

Julibrine I	Structural Classification Natural Products Albizia julibrissin Durazz. Leguminosae Source classification Plants	Others
Julibrine I is a pyridoxine derivative found in the fresh stem bark of Albizzia julibrissin DURAzz, IV .

HY-125676

Thermopterin	Structural Classification Natural Products Microorganisms Source classification	Drug Derivative Bacterial
Thermopterin is a derivative of the antimicrobial agent Pterin (HY-W037825) isolated from Methanoculleus thermophilus .

HY-N11789

3-Hydroxyirisquinone	Quinones Structural Classification Iridaceae Source classification Benzene Quinones Plants Iris bungei Maxim.	Others
3-Hydroxyirisquinone is a quinone derivative, which can isolated from the seeds of Iris bungei Maxim .

HY-134663

2-O-β-D-Glucosyloxy-4-methoxybenzene propanoic acid	Structural Classification Ketones, Aldehydes, Acids Labiatae Source classification Peucephyllum schottii A.Gray Plants	Others
2-O-β-D-Glucosyloxy-4-methoxybenzene propanoic acid is a glucoside derivative .

HY-126126

S-Adenosyl-DL-methionine	Structural Classification Classification of Application Fields Ketones, Aldehydes, Acids Source classification Other Diseases Endogenous metabolite Disease Research Fields	Drug Derivative
S-Adenosyl-DL-methionine is a derivative of Ademetionine (HY-B0617). Ademetionine is an intermediate metabolite of methionine .

HY-Y1139

Pimelic acid 2 Publications Verification Heptanedioic acid; 1,5-Pentanedicarboxylic acid; 1,7-Heptanedioic acid	Structural Classification Immune System Disorder Microorganisms Classification of Application Fields Ketones, Aldehydes, Acids Source classification Disease markers Metabolic Disease Endogenous metabolite Disease Research Fields	Endogenous Metabolite
Pimelic acid is the organic compound and its derivatives are involved in the biosynthesis of the amino acid called lysine.Pimelic acid can be used in keratoconus research .

HY-119543

O-Succinyl-L-homoserine	Human Gut Microbiota Metabolites Microorganisms Source classification Endogenous metabolite	Amino Acid Derivatives
O-Succinyl-L-homoserine is a homoserine derivative. O-Succinyl-L-homoserine is an intermediate in the biosynthesis of methionine in Escherichia coli and Salmonella typhimurium .

HY-N11791

Qianhucoumarin B	Structural Classification Chrysanthemum × morifolium (Ramat.) Hemsl. Source classification Coumarins Phenylpropanoids Plants Umbelliferae	Others
Qianhucoumarin B is a coumarin derivative. Qianhucoumarin B can be isolated from from the traditional Chinese medicine Qianhu, roots of Peucedanum praeruptorum .

HY-19355

Rocagloic acid	Structural Classification Classification of Application Fields Ketones, Aldehydes, Acids Source classification Plants Meliaceae Disease Research Fields Aglaia elliptifolia Cancer	Others
Rocagloic acid is a racaglamide derivative isolated from the fruits of Aglaia elliptifolia with potent cytotoxicity .

HY-N3198A

Sophoramine (-)-Sophoramine	Alkaloids Classification of Application Fields Leguminosae Source classification Other Diseases Pyridine Alkaloids Plants Sophora flavescens Aiton Disease Research Fields	Others
Sophoramine ((-)-Sophoramine), an alkaloid, is a dehydro-derivative of Matrine .

HY-N2857

Alpinumisoflavone	Flavonoids Classification of Application Fields Leguminosae Source classification Other Diseases Phenols Polyphenols Plants Disease Research Fields Isoflavones Erythrina variegata Linn.	Others
Alpinumisoflavone (compound 2) is a flavonoid derivative isolated from the stem bark of Erythrina lysistemon Hutch .

HY-N0947R

(-)-Anomalin (Standard)	Structural Classification Source classification Coumarins Salvia hypargeia Fisch. & C.A.Mey. Phenylpropanoids Umbelliferae Plants Artemisia vulgaris L.	Others
(-)-Anomalin (Standard) is the analytical standard of (-)-Anomalin. This product is intended for research and analytical applications. (-)-Anomalin ((-)-Praeruptorin B) is a coumarin derivative isolated from the root of Angelica anomala .

HY-N12471

Gossypetin 3′-O-glucoside	Malvaceae Structural Classification Flavonols Flavonoids Source classification Plants Hibiscus elatus Sw.	Others
Gossypetin 3′-O-glucoside is a gossypetin derivative. Gossypetin 3′-O-glucoside can be isolated from ethanolic extracts after Soxhlet extraction .

HY-N12350

Ellagic acid 3-O-α-L-rhamnopyranoside	Structural Classification Flavonoids Staphyleaceae Source classification Plants Biflavones Turpinia arguta (Lindl.) Seem.	Others
Ellagic acid 3-O-α-L-rhamnopyranoside is an ellagic acid derivative can be isolated from Folium Turpiniae .

HY-N11993

Aloveroside A	Structural Classification Polysaccharides Liliaceae Source classification Aloe vera (L.) Burm. f. Plants Saccharides	Cholinesterase (ChE)
Aloveroside A is a triglucosylnaphthalene derivative isolated from ethanolic extract of aloe vera. Aloveroside A has weak bACE inhibitory activity (inhibition rate at a dose of 100 μg/mL is approximately 18.68%) .

HY-N10752

6,7-Dihydroxy-2-(2-phenylethyl)-5,6,7,8-tetrahydrochromone	Structural Classification Natural Products Thymelaeaceae Source classification Plants Aquilaria sinensis (Lour.) Spreng.	Others
6,7-Dihydroxy-2-(2-phenylethyl)-5,6,7,8-tetrahydrochromone is a natural chromone derivative found in withered wood of Aquilaria sinensis .

HY-N0572

9-Hydroxycamptothecin 9-Hydroxycamptothecine	Alkaloids Structural Classification Monophenols Classification of Application Fields Source classification Phenols Camptotheca acuminata Decne. Nyssaceae Plants Disease Research Fields Indole Alkaloids Cancer	Drug Derivative
9-Hydroxycamptothecin (9-Hydroxycamptothecine; compound 23c) is a Camptothecin (HY-16560) derivative with anticancer activities .

HY-W008642

Leu-Leu-OH L-Leucyl-L-leucine	Natural Products Classification of Application Fields Source classification Other Diseases Endogenous metabolite Disease Research Fields	Amino Acid Derivatives
Leu-Leu-OH (L-Leucyl-L-leucine), a Leu derivative, is a neutral dipeptide that can be used to study the functionality of dileucine motifs .

HY-Y1139R

Pimelic acid (Standard)	Structural Classification Immune System Disorder Microorganisms Ketones, Aldehydes, Acids Source classification Disease markers Endogenous metabolite	Endogenous Metabolite
Pimelic acid (Standard) is the analytical standard of Pimelic acid. This product is intended for research and analytical applications. Pimelic acid is the organic compound and its derivatives are involved in the biosynthesis of the amino acid called lysine.Pimelic acid can be used in keratoconus research .

HY-N8344

Frangulin A	Ventilago leiocarpa Benth. Quinones Structural Classification Anthraquinones Source classification Plants Rhamnaceae	Others
Frangulin A is a emodin derivative. Frangulin A can be obtained from Ventilago leiocarpa Benth .

HY-N3263

Methyleugenolglycol	Structural Classification Natural Products Classification of Application Fields Source classification Other Diseases Endogenous metabolite Disease Research Fields	Others
Methyleugenolglycol (Compound XIV) is a metabolism of alkenebenzene derivative .

HY-N1854

Pinobanksin 3-acetate	Flavanonols Structural Classification Flavonoids Animals Classification of Application Fields Other Diseases Scrophulariaceae Eremophila alternifolia Plants Disease Research Fields	Others
Pinobanksin 3-acetate is a one of Pinobanksin ester derivatives that can be isolated from Sonoran propolis .

HY-N7724

Cedrusin (+)-Cedrusin	Styrax suberifolius Hook. et Arn. Source classification Styracaceae Plants	Others
Cedrusin is a benzofuran derivative that can be isolated from Styrax suberifolius .

HY-N10077

Eriosemation Lupichromone	Structural Classification Natural Products Leguminosae Flemingia philippinensis Merr. et Rolfe Source classification Phenols Polyphenols Plants	Others
Eriosemation is a chromone derivatives that can be isolated from Flemingia philippinensis .

HY-133860

Chrysoobtusin	Seeds of Cassia tora Linn. Structural Classification Classification of Application Fields Source classification Plants Quinones other families Leguminosae Anthraquinones Other Diseases Phenols Polyphenols Disease Research Fields	Drug Derivative
Chrysoobtusin is an anthraquinone derivative isolated from Semen Cassiae. Semen Cassiae has long been used to protect liver, brighten eyes, and relieve constipation .

HY-N1800

3,3'-Di-O-methylellagic acid-4'-O-β-D-glucopyranoside	Structural Classification Monophenols Classification of Application Fields Ketones, Aldehydes, Acids Source classification Celastraceae Other Diseases Phenols Plants Disease Research Fields Dipentodon sinicus Dunn	Others
3,3'-Di-O-methylellagic acid-4'-O-β-D-glucopyranoside is a ellagic acid derivative that can be isolated from Dipentodon sinicus .

HY-N13086

Peniviridiol A	Structural Classification Microorganisms Terpenoids Sesquiterpenes Source classification	Others
Peniviridiol A (compound4) is a viridin derivative that can be isolated from rhizosphere fungus Penicillium sp. SMU0102 .

HY-N3045

(S,S)-Pisatin	Natural Products Classification of Application Fields Leguminosae Source classification Other Diseases Pisum sativum Linn Plants Disease Research Fields	Others
(S,S)-Pisatin (compound 8) is a dimeric pterocarpan derivative is isolated from the grains of millettia pachyloba .

HY-N1069

Wittifuran X	Structural Classification Source classification Phenols Polyphenols Morus wittiorum Hand.-Mazz. Plants Moraceae	Others
Wittifuran X is a 2-arylbenzofuran derivative, which can be isolated from the stem bark of Morus wittiorum .

HY-113225

Guanosine triphosphate GTP	Infection Structural Classification Natural Products Classification of Application Fields Source classification Endogenous metabolite Disease Research Fields Cancer	SARS-CoV Nucleoside Antimetabolite/Analog DNA/RNA Synthesis Endogenous Metabolite
Guanosine triphosphate is a native nucleotide. The derivatives of GTP may be used as specific inhibitors against COVID-19 .

HY-N7889

Syringetin-3-O-rutinoside	Flavonols Flavonoids Classification of Application Fields Larix sibirica Ledeb. Pinaceae Source classification Other Diseases Phenols Polyphenols Plants Disease Research Fields	Others
Syringetin-3-O-rutinoside is an antioxidant compound . Syringetin-3-O-rutinoside can be used for the synthesis of syringetin-O-glycoside derivatives .

HY-N12801

3-Hydroxy-1,2-dimethoxyxanthone	Structural Classification Xanthones Polygala nitida Source classification Polygalaceae Phenols Plants	Others
3-Hydroxy-1,2-dimethoxyxanthone is a xanthone derivative and can be isolated from Polygala nitida .

HY-N10200

2,7-Dimethoxy-6-(1-acetoxyethyl)juglone	Quinones Monophenols Microorganisms Classification of Application Fields Anthraquinones Source classification Other Diseases Phenols Disease Research Fields	Others
2,7-Dimethoxy-6-(1-acetoxyethyl)juglone is a naphthoquinone derivative found in the fungus Kirschsteiniothelia species .

HY-N11978

6-Hydroxykynurenic acid 6-HKA	Structural Classification Ginkgoaceae Ketones, Aldehydes, Acids Source classification Plants Ginkgo biloba	iGluR
6-Hydroxykynurenic acid (6-HKA) is a derivative of kynurenic acid (KYNA) and can be isolated from Ginkgo leaves. 6-Hydroxykynurenic acid is a low-affinity NMDAR antagonist (IC₅₀: 59 μM) .

HY-N10007

Dodoviscin J	Structural Classification Flavonoids Flavones Dodonaea viscosa (L.) Jacq. Source classification Sapindaceae Plants	Others
Dodoviscin J is a prenyl flavonol derivative can be isolated from the aerial parts of Dodonaea viscosa .

HY-121184

Epicoccamide	Alkaloids Microorganisms Pyrrole Alkaloids Classification of Application Fields Source classification Other Diseases Disease Research Fields	Endogenous Metabolite
Epicoccamide, a tetramic acid derivative, is secondary metabolite from Epicoccum purpurascens .

HY-I0960

Uracil 3 Publications Verification	Structural Classification Natural Products Human Gut Microbiota Metabolites Microorganisms Classification of Application Fields Disease markers Endocrine diseases Nervous System Disorder Endogenous metabolite Disease Research Fields Cancer	Endogenous Metabolite Drug Derivative
Uracil is a pyrimidine derivative and one of the four nucleobases in the nucleic acid of RNA. Uracil is a frequently occurring DNA base damage that results from the spontaneous or chemically induced deamination of cytosine and is mutagenic at the level of replication. Uracil could potentially alter transcriptional fidelity, resulting in production of mutant proteins .

HY-N10925

9-Hydroxythymol	Structural Classification Other Monoterpenes Glycyrrhiza pallidiflora Maxim. Terpenoids Source classification Phenols Plants Compositae	Others
9-Hydroxythymol is a thymol derivative. 9-Hydroxythymol can be isolated from Eupatorium fortunei .

Cat. No.	Product Name	Chemical Structure

HY-14273S

Isavuconazole-d4
Isavuconazole-d₄ is a deuterium labeled Isavuconazole (BAL-4815). Isavuconazole is a triazole proagent with antifungal activity against yeasts, molds, and dimorphic fungi[1].

HY-Y0688S

1H-Benzotriazole-4,5,6,7-d4
1H-Benzotriazole-4,5,6,7-d₄ is the deuterium labeled 1H-Benzo[d][1,2,3]triazole[1].

HY-17373S

Posaconazole-d5
Posaconazole-d₅ is a deuterium-labeled form of Posaconazole. Posaconazole is a broad-spectrum, second generation, triazole compound with antifungal activity[1].

HY-17373S1

Posaconazole-d4
Posaconazole-d₄ is a deuterium-labeled form of Posaconazole. Posaconazole is a broad-spectrum, second generation, triazole compound with antifungal activity[1].

HY-12772S

Hydroxy Itraconazole-d8
Hydroxy Itraconazole-d₈ is the deuterium labeled Hydroxy Itraconazole. Hydroxy Itraconazole is an active metabolite of Itraconazole (ITZ), which is a triazole antifungal agent.

HY-141941S

Triazole Lactic Acid-13C2, 15N3
Triazole Lactic Acid- ¹³C₂, ¹⁵N₃ is the ¹³C and ¹⁵N labeled Triazole Lactic Acid[1].

HY-W098127S

*Methyl 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxylate-d2*
Methyl 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxylate-d₂ is the deuterium labeled Methyl 1-(2,6-difluorobenzyl)-1H-1,2,3-triazole-4-carboxylate[1].

HY-Y0219S1

*1,2,4-Triazole-d3*
NSC 83128-d₃ is the deuterium labeled NSC 83128[1].

HY-W705791

Metconazole-d6
Metconazole-d₆ is the deuterium labeled Metconazole. Metconazole is a triazole fungicide agent.

HY-W749242

Paclobutrazol-d4
Paclobutrazol-d₄ is the deuterium labeled Paclobutrazol. Paclobutrazol is a triazole-containing plant growth retardant that is known to inhibit the biosynthesis of gibberellins .

HY-113225S2

Guanosine triphosphate-13C dilithium
Guanosine triphosphate- ¹³C (GTP- ¹³C) dilithium is ¹³C-labeled Guanosine triphosphate (HY-113225). Guanosine triphosphate is a native nucleotide. The derivatives of GTP may be used as specific inhibitors against COVID-19.

HY-113225S3

Guanosine triphosphate-15N5 dilithium
Guanosine triphosphate- ¹⁵N₅ (GTP- ¹⁵N₅) dilithium is ¹⁵N labeled Guanosine triphosphate (HY-113225). Guanosine triphosphate is a native nucleotide. The derivatives of GTP may be used as specific inhibitors against COVID-19.

HY-113225S5

Guanosine triphosphate-13C10 dilithium
Guanosine triphosphate- ¹³C₁₀ (GTP- ¹³C₁₀) dilithium is ¹³C-labeled Guanosine triphosphate (HY-113225). Guanosine triphosphate is a native nucleotide. The derivatives of GTP may be used as specific inhibitors against COVID-19.

HY-17373S3

Posaconazole-d7
Posaconazole-d₇ (SCH 56592-d₇) is deuterium labeled Posaconazole. Posaconazole is a broad-spectrum, second generation, triazole compound with antifungal activity.

HY-17373S2

Posaconazole-d3
Posaconazole-d₃ (SCH 56592-d₃) is deuterium labeled Posaconazole. Posaconazole is a broad-spectrum, second generation, triazole compound with antifungal activity.

HY-B0851S

Triadimenol-d4
Triadimenol-d₄ is the deuterium labeled Triadimenol[1]. Triadimenol is a triazole fungicide and has been widely used in agriculture. Triadimenol has certain toxicity to animals[2].

HY-113225S4

Guanosine triphosphate-15N5,d14 dilithium
Guanosine triphosphate- ¹⁵N₅,d₁₄ (GTP- ¹⁵N₅,d₁₄) dilithium is deuterium and ¹⁵N labeled Guanosine triphosphate (HY-113225). Guanosine triphosphate is a native nucleotide. The derivatives of GTP may be used as specific inhibitors against COVID-19.

HY-Y0302S

Diammonium phosphate-15N2
Diammonium phosphate- ¹⁵N₂ is ¹⁵N₂ labeled Diammonium phosphate (HY-Y0302). Diammonium phosphate is a neutral and efficient catalyst in 1,8-Dioxo-octahydroxanthene derivatives synthesis, which can be used as an excipient, such as diuretic, buffer, effervescent .

HY-136457S

2-NP-AHD-13C3
2-NP-AHD- ¹³C₃ is the ¹³C labled 2-NP-AHD (HY-136457) . 2-NP-AHD is a 2-nitrophenyl derivative of AHD (a metabolite of nitrofurans type of antibiotics), can be used as indicator of the illegal usage of nitrofuran agents .

HY-Y0219S

*1,2,4-Triazole-13C2,15N3*
NSC 83128- ¹³C₂, ¹⁵N₃ is the ¹³C and ¹⁵N labeled NSC 83128[1].

HY-12772S3

Hydroxy Itraconazole-d6
Hydroxy Itraconazole-d₆ (R-63373-d₆) is deuterium labeled Hydroxy Itraconazole. Hydroxy Itraconazole (Itraconazole metabolite Hydroxy Itraconazole; R-63373) is an active metabolite of Itraconazole (ITZ), which is a triazole antifungal agent.

HY-135761S

Penconazole-d7
Penconazole-d₇ is the deuterium labeled Penconazole[1]. Penconazole is a typical triazole fungicide, and mainly applied on apples, grapes, and vegetables to control powdery mildew. Penconazole inhibits sterol biosynthesis in fungi. Penconazole decrease AChE activity in the cerebrum and cerebellum of rats[2][3].

HY-76200S

Voriconazole-d3
Voriconazole-d₃ is the deuterium labeled Voriconazole. Voriconazole (UK-109496) is a second-generation, broad-spectrum triazole antifungal agent that inhibits fungal ergosterol biosynthesis. Voriconazole exerts its antifungal activity by inhibition of 14-α-lanosterol demethylation, which is mediated by fungal cytochrome P450 enzymes[1][2].

HY-B0101S

Fluconazole-d4
Fluconazole-d₄ is the deuterium labeled Fluconazole. Fluconazole (UK-49858) is a triazole antifungal agent with excellent activities against a broad range of fungi, especially against Candida albicans. Fluconazole inhibits C. albicans and Candida kefyr with IC99s range from 0.20 μg/mL to 0.39 μg/mL[1].

HY-W706180

(±)-Triadimefon-d4

(±)-Triadimefon-d₄ is deuterium labeled Triadimefon. Triadimefon is a triazole fungicide used to control powdery mildew, rusts, and other fungal pests on grains, fruit and vegetable crops, turf, shrubs, and trees. Triadimefon inhibits lanosterol 14α-demethylase, interfering with oxidative demethylation reactions in the ergosterol biosynthesis pathway of fungi, and also blocks gibberellin biosynthesis .

HY-144378S

*Thiorphan methoxyacetophenone derivative-d7*
Thiorphan methoxyacetophenone derivative-d₇ is the deuterium labeled Thiorphan methoxyacetophenone derivative[1].

HY-15660S

Efinaconazole-d4
Efinaconazole-d₄ is the deuterium labeled Efinaconazole. Efinaconazole (KP-103) is a triazole antifungal agent and againsts T. mentagrophytes SM-110 and C. albicans ATCC 10231 with MICs of 0.0039 μg/mL and 0.00098 μg/mL, respectively[1]. Efinaconazole has a potent in vitro activity against fungal pathogens including dermatophytes, Candida and Malassezia species[1].

HY-17514S

Itraconazole-d5

Itraconazole-d₅ is the deuterium labeled Itraconazole. Itraconazole (R51211) is a triazole antifungal agent and a potent and orally active Hedgehog (Hh) signaling pathway antagonist with an IC50 of ~800 nM. Itraconazole potently inhibits lanosterol 14α-demethylase (cytochrome P450 enzyme), thereby inhibits the oxidative conversion of lanosterol to ergosterol. Itraconazole has anticancer and antiangiogenic effects[1][2][3].

HY-Z2483S

*Clopidogrel-MP endo derivative-13C,d3*
Clopidogrel-MP endo derivative- ¹³C,d₃ is the deuterium and ¹³C labeled Clopidogrel-MP endo derivative[1].

HY-17514S2

Itraconazole-d9

Itraconazole-d₉ is the deuterium labeled Itraconazole[1]. Itraconazole (R51211) is a triazole antifungal agent and a potent and orally active Hedgehog (Hh) signaling pathway antagonist with an IC50 of ~800 nM. Itraconazole potently inhibits lanosterol 14α-demethylase (cytochrome P450 enzyme), thereby inhibits the oxidative conversion of lanosterol to ergosterol. Itraconazole has anticancer and antiangiogenic effects. Itraconazole is a oxysterol-binding protein (OSBP) inhibitor[2][3][4][5].

HY-20582S

L-Prolinamide-d3
L-Prolinamide-d₃ is the deuterium labeled L-Prolinamide[1]. L-Prolinamide is a proline derivative[2].

HY-B0101S1

Fluconazole-13C2,15N
Fluconazole-13C2,15N (UK-49858-13C2,15N) is the ¹³C and ¹⁵N labeled isotope of Fluconazole (HY-B0101). Fluconazole (UK-49858) is a triazole antifungal agent with excellent activities against a broad range of fungi, especially against Candida albicans. Fluconazole inhibits C. albicans and Candida kefyr with IC₉₉s range from 0.20 μg/mL to 0.39 μg/mL .

HY-79131S5

Fmoc-Phe-OH-13C
Fmoc-Phe-OH- ¹³C is the ¹³C labeled Fmoc-Phe-OH[1]. Fmoc-Phe-OH is a phenylalanine derivative[2].

HY-W037443S

Methyl L-valinate-d8
Methyl L-valinate-d₈ is the deuterium labeled Methyl L-valinate[1]. Methyl L-valinate is a valine derivative[2].

HY-13566AS

Belotecan-d7 hydrochloride
Belotecan-d₇ (hydrochloride) is the deuterium labeled Belotecan hydrochloride. Belotecan hydrochloride (CKD-602 hydrochloride), a Topoisomerase I inhibitor, is a synthetic camptothecin derivative[1][2].

HY-113411S

3-Hydroxyglutaric acid-d5
3-Hydroxyglutaric acid-d₅ is the deuterium labeled 3-Hydroxyglutaric acid. 3-Hydroxyglutaric acid is a glutaric acid derivative[1][2].

HY-B0847S1

Propiconazole-d3 nitrate

Propiconazole-d₃ (nitrate) is the deuterium labeled Propiconazole nitrate. Propiconazole is a broad-spectrum triazole fungicide that inhibits the conversion of lanosterol to ergosterol, leading to fungal cell membrane disruption. Propiconazole inhibits S. cerevisiae, but not rat liver, microsomal cytochrome P450 (IC50s=0.04 and >200 µM, respectively). Propiconazole inhibits the growth of T. deformans and R. stolonifer (ED50s=0.073 and 4.6 µg/mL, respectively). Propiconazole increases production of reactive oxygen species (ROS).

HY-B0847S

Propiconazole-d7

Propiconazole-d₇ is the deuterium labeled Propiconazole. Propiconazole is a broad-spectrum triazole fungicide that inhibits the conversion of lanosterol to ergosterol, leading to fungal cell membrane disruption. Propiconazole inhibits S. cerevisiae, but not rat liver, microsomal cytochrome P450 (IC50s=0.04 and >200 µM, respectively). Propiconazole inhibits the growth of T. deformans and R. stolonifer (ED50s=0.073 and 4.6 µg/mL, respectively). Propiconazole increases production of reactive oxygen species (ROS)[1].

HY-W007941S1

Fmoc-Ser(tBu)-OH-15N
Fmoc-Ser(tBu)-OH- ¹⁵N is the ¹⁵N labeled Fmoc-Ser(tBu)-OH[1]. Fmoc-Ser(tBu)-OH is a serine derivative[2].

HY-16760S

9-cis-Retinol acetate-d5
9-cis-Retinol acetate-d₅ is the deuterium labeled 9-cis-Retinol acetate. 9-cis-Retinol acetate is a retinal derivative[1][2].

HY-W007798S1

Fmoc-Cys(Trt)-OH-d2
Fmoc-Cys(Trt)-OH-d₂ is the deuterium labeled Fmoc-Cys(Trt)-OH. Fmoc-Cys(Trt)-OH is an N-terminal protected cysteine derivative[1].

HY-19821S1

Fmoc-Ile-OH-13C6,15N
Fmoc-Ile-OH- ¹³C₆, ¹⁵N is the ¹³C and ¹⁵N labeled Fmoc-Ile-OH[1]. Fmoc-Ile-OH is an isoleucine derivative[2].

HY-W012497S

N-Acetyl-D-methionine-d4
N-Acetyl-D-methionine-d₄ is the deuterium labeled N-Acetyl-D-methionine[1]. N-Acetyl-D-methionine is a Methionine (HY-13694) derivative[2].

HY-116666S

(Rac)-Etomidate acid-d5
Nonanoic acid-d2 is the deuterium labeled (Rac)-Etomidate acid .

HY-Y1838S

Methoxytrimethylsilane-d3
Methoxytrimethylsilane-d₃ is the deuterium labeled Methoxytrimethylsilane. Methoxytrimethylsilane is a mono-alkoxy derivative .

HY-158995S

3-Epiglycyrrhetinic acid-d2
3-Epiglycyrrhetinic acid-d2 (3α-Glycyrrhetic acid-d2) is the deuterium-labeled 3-Epiglycyrrhetinic acid. 3-Epiglycyrrhetinic acid is a derivative of glycyrrhetic acid. Glycyrrhetic acid and its derivative are considered to have anti-inflammatory, anti-ulcer, and antiviral activities .

HY-158995S1

3-Epiglycyrrhetinic acid-d3
3-Epiglycyrrhetinic acid-d3 (3α-Glycyrrhetic acid-d3) is the deuterium-labeled 3-Epiglycyrrhetinic acid. 3-Epiglycyrrhetinic acid is a derivative of glycyrrhetic acid. Glycyrrhetic acid and its derivative are considered to have anti-inflammatory, anti-ulcer, and antiviral activities .

HY-W014375S3

Arginine-d7 hydrochloride
Arginine-d₇ hydrochloride is deuterium labeled Arginine (hydrochloride) (HY-W014375). Arginine hydrochloride is an arginine derivative.

HY-113404S

DL-Dopa-d6
DL-Dopa-d₆ is the deuterium labeled DL-Dopa. DL-Dopa is a beta-hydroxylated derivative of phenylalanine.

HY-79096S

BOC-L-Phenylalanine-13C
BOC-L-Phenylalanine- ¹³C is a ¹³C-labeled BOC-L-Phenylalanine. BOC-L-Phenylalanine is a derivative of Phenylalanine[1].

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